SCHEMBL4785757

SCHEMBL4785757

CN1CCC(Oc2nc(-c3cccc(O)c3)nc(N3Cc4ccccc4C[C@@H]3CO)n2)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 8/20 0.36
PIK3R1 P27986 1/20 0.36
ADORA3 P0DMS8 1/20 0.35
ADORA1 P30542 1/20 0.35
MET P08581 1/20 0.34
CHEK1 O14757 1/20 0.34
JAK2 O60674 1/20 0.34
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
CHRM3 P20309 2/20 0.33
ESRRG P62508 1/20 0.33
IDH1 O75874 1/20 0.33
HSD17B2 P37059 1/20 0.33
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
CHRM5 P08912 1/20 0.32
CHRM1 P11229 1/20 0.32
SCN1A P35498 1/20 0.32
SCN2A Q99250 1/20 0.32
SCN3A Q9NY46 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14161674 0.96 PIK3CA (0.35) PIK3CAPIK3R1ADORA3ADORA1MET
SCHEMBL4784163 0.96 PIK3CA (0.35) PIK3CAPIK3R1ADORA3ADORA1MET
SCHEMBL4785566 0.92 CHRM3 (0.35) PIK3CAPIK3R1ADORA3ADORA1CHRM3
SCHEMBL14161656 0.89 PIK3CA (0.40) PIK3CAPIK3R1MTOR
SCHEMBL14161859 0.86 PIK3CA (0.38) PIK3CAPIK3R1CHEK1MTOR
SCHEMBL4781444 0.83 PIK3CA (0.35) PIK3CAPIK3R1ADORA3ADORA1CHEK1
SCHEMBL4783926 0.83 HRH4 (0.44) PIK3CAPIK3R1ADORA3ADORA1MTOR
SCHEMBL4846093 0.83 HRH4 (0.44) PIK3CAPIK3R1ADORA3ADORA1MTOR
SCHEMBL4785845 0.83 HRH4 (0.44) PIK3CAPIK3R1ADORA3ADORA1MTOR
SCHEMBL4784229 0.82 PIK3CA (0.35) PIK3CAPIK3R1CHEK1JAK2MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008072850-A1 TRIAZINE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST ACETYL-COA CARBOXYLASE AMOREPACIFIC CORPORATION (KR) 2008-06-19 WO disclosed