SCHEMBL4786332

SCHEMBL4786332

Cc1nc(-c2ccc(Cl)cc2)c(C(=O)N2CCC[C@H]2CNC(=O)c2c(C)nc3sccn23)s1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 14/20 0.51
HCRTR2 O43614 11/20 0.51
NR1I3 Q14994 1/20 0.43
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
MAPK1 P28482 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1398754 0.95 HCRTR1 (0.53) HCRTR1HCRTR2NR1I3
SCHEMBL4743875 0.91 HCRTR1 (0.53) HCRTR1HCRTR2
SCHEMBL4740957 0.90 HCRTR1 (0.54) HCRTR1HCRTR2
SCHEMBL4741690 0.90 HCRTR1 (0.54) HCRTR1HCRTR2
SCHEMBL1398768 0.89 HCRTR1 (0.56) HCRTR1HCRTR2
SCHEMBL1398798 0.88 HCRTR1 (0.53) HCRTR1HCRTR2
SCHEMBL1398771 0.87 HCRTR1 (0.52) HCRTR1HCRTR2
SCHEMBL4739904 0.87 HCRTR1 (0.53) HCRTR1HCRTR2
SCHEMBL1398725 0.86 HCRTR1 (0.58) HCRTR1HCRTR2
SCHEMBL4739191 0.86 HCRTR1 (0.52) HCRTR1HCRTR2KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008087611-A2 PYRROLIDINE- AND PIPERIDINE- BIS-AMIDE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2008-07-24 WO disclosed