SCHEMBL4786548

SCHEMBL4786548

CC(C)c1cc(-c2nnc(O)n2-c2ccc(N(C)C)c(F)c2)c(O)cc1O

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 20/20 0.55
HSP90AB1 P08238 20/20 0.55
HSP90B1 P14625 1/20 0.38
TRAP1 Q12931 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4786259 0.88 HSP90AA1 (0.48) HSP90AA1HSP90AB1
Hydrochloric Acid SCHEMBL4787381 0.87 HSP90AA1 (0.47) HSP90AA1HSP90AB1
SCHEMBL1304307 0.83 HSP90AA1 (0.71) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL4786852 0.82 HSP90AA1 (0.78) HSP90AA1HSP90AB1
Hydrochloric Acid SCHEMBL1304868 0.82 HSP90AA1 (0.70) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL12060284 0.79 HSP90AA1 (0.63) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL1304392 0.79 HSP90AA1 (0.67) HSP90AA1HSP90AB1
Hydrochloric Acid SCHEMBL1304249 0.78 HSP90AA1 (0.66) HSP90AA1HSP90AB1
SCHEMBL4743521 0.77 HSP90AA1 (0.57) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL14777477 0.77 HSP90AA1 (0.57) HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008103353-A1 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY SYNTA PHARMACEUTICALS CORP. (US) 2008-08-28 WO claimed
WO-2008103353-A1 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY SYNTA PHARMACEUTICALS CORP. (US) 2008-08-28 WO disclosed