SCHEMBL4787966

SCHEMBL4787966

CN(C(=O)OC(C)(C)C)c1cccc(CCCc2ccc(C[C@H](NC(=O)OC(C)(C)C)C(=O)O)s2)n1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 3/20 0.49
ITGA5 P08648 3/20 0.49
ITGAV P06756 2/20 0.49
ITGB3 P05106 2/20 0.49
CTSS P25774 6/20 0.40
CTSK P43235 6/20 0.40
ACE P12821 1/20 0.39
PTPN1 P18031 2/20 0.39
ITGB6 P18564 1/20 0.38
ITGA2B P08514 1/20 0.37
SCN9A Q15858 1/20 0.37
PPARA Q07869 4/20 0.36
PPARG P37231 3/20 0.36
ITGA4 P13612 1/20 0.35
ITGB7 P26010 1/20 0.35
CTSL P07711 1/20 0.35
PPARD Q03181 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4064751 0.93 ITGAV (0.42) ITGB1ITGA5ITGAVITGB3CTSS
SCHEMBL4940782 0.83 PTPN1 (0.39) ITGB1ITGA5ITGAVITGB3CTSS
SCHEMBL4940785 0.83 PTPN1 (0.39) ITGB1ITGA5ITGAVITGB3CTSS
SCHEMBL4074572 0.80 KLK5 (0.44) ITGB1ITGA5ITGB3CTSSCTSK
SCHEMBL4788504 0.78 ITGAV (0.46) ITGB1ITGA5ITGAVITGB3CTSS
SCHEMBL8228529 0.78 KLK5 (0.44) ITGB1ITGA5ITGB3CTSSCTSK
SCHEMBL4067205 0.78 KLK5 (0.44) ITGB1ITGA5ITGB3CTSSCTSK
SCHEMBL4070076 0.77 KLK5 (0.35) CTSSCTSKPTPN1SCN9ACTSL
SCHEMBL4070078 0.77 KLK5 (0.35) CTSSCTSKPTPN1SCN9ACTSL
SCHEMBL4069200 0.76 ITGB1 (0.43) ITGB1ITGA5ITGB3CTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008125811-A1 N-[HETEROARYLCARBONYL]-S-THIENYL-L-ALANINE DERIVATIVES AS α5β1 ANTAGONISTS ASTRAZENECA AB (SE) 2008-10-23 WO disclosed