SCHEMBL4789570

SCHEMBL4789570

C[C@@H](NN(C[C@H]1CN(C(=O)c2ccc(S(N)(=O)=O)cc2)C[C@@H]1c1ccccc1)C(=O)O)c1cccc2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CASR P41180 5/20 0.46
CYP2D6 P10635 2/20 0.42
CA1 P00915 9/20 0.41
CA2 P00918 9/20 0.41
CA9 Q16790 9/20 0.41
CA12 O43570 5/20 0.41
CA7 P43166 4/20 0.41
CA14 Q9ULX7 3/20 0.41
CCR5 P51681 3/20 0.39
CA4 P22748 4/20 0.39
TLR2 O60603 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4108723 0.87 CA1 (0.43) CASRCYP2D6CA1CA2CA9
SCHEMBL4106554 0.86 CASR (0.49) CASRCYP2D6CA1CA2CA9
SCHEMBL4106558 0.86 CASR (0.49) CASRCYP2D6CA1CA2CA9
SCHEMBL4789572 0.82 CA1 (0.43) CASRCYP2D6CA1CA2CA9
SCHEMBL4106863 0.76 SCN3A (0.42) CASRCYP2D6CCR5TLR2
SCHEMBL4106204 0.75 CCR5 (0.44) CASRCYP2D6CCR5TLR2
SCHEMBL4100239 0.74 CCR5 (0.41) CASRCYP2D6CCR5TLR2
Hydrochloric Acid SCHEMBL4106570 0.74 CASR (0.54) CASRCYP2D6CCR5
SCHEMBL4094857 0.73 CASR (0.51) CASRCYP2D6CCR5TLR2
SCHEMBL4094852 0.73 CASR (0.51) CASRCYP2D6CCR5TLR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1882684-A1 PYRROLIDINE DERIVATIVE OR SALT THEREOF Astellas Pharma Inc. (JP) 2008-01-30 EP disclosed