SCHEMBL4789733

SCHEMBL4789733

c1ccc(-c2cc(CN3CCCC3)ccn2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.57
TGFBR1 P36897 1/20 0.51
CXCR4 P61073 2/20 0.49
CYP2D6 P10635 2/20 0.47
CYP2C19 P33261 1/20 0.47
DRD2 P14416 1/20 0.47
DRD4 P21917 1/20 0.47
DRD3 P35462 1/20 0.47
CYP2C9 P11712 1/20 0.47
HIF1A Q16665 1/20 0.47
TSHR P16473 2/20 0.46
ALDH1A1 P00352 1/20 0.46
HTR1A P08908 2/20 0.45
HTR7 P34969 2/20 0.45
PRMT6 Q96LA8 1/20 0.45
CHRNB2 P17787 1/20 0.45
CHRNA4 P43681 1/20 0.45
HCRTR1 O43613 2/20 0.45
HCRTR2 O43614 2/20 0.45
ASIC3 Q9UHC3 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29204486 0.84 DRD2 (0.45) KDRCXCR4DRD2DRD4DRD3
SCHEMBL10375716 0.83 MEN1 (0.55) DRD2DRD4DRD3
SCHEMBL6057472 0.82 CXCR4 (0.57) KDRTGFBR1CXCR4CYP2D6CYP2C9
SCHEMBL10373762 0.81 OPRL1 (0.62) DRD2DRD4DRD3ALDH1A1
Hydrochloric Acid SCHEMBL7958693 0.81 CCR3 (0.61) DRD2DRD4DRD3ALDH1A1SMN1; SMN2
SCHEMBL10374922 0.80 DRD4 (0.54) DRD2DRD4DRD3TSHRALDH1A1
SCHEMBL10374834 0.79 HTR2A (0.53) DRD2DRD4DRD3CYP2C9ALDH1A1
SCHEMBL7161609 0.79 HCRTR1 (0.51) DRD2DRD4DRD3CYP2C9ALDH1A1
SCHEMBL10373580 0.78 MEN1 (0.62) DRD2DRD4DRD3ALDH1A1
SCHEMBL10374924 0.78 DRD2 (0.47) DRD2DRD4DRD3HTR1AHCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902025-A1 KINASE INHIBITORS Allergan, Inc. (US) 2008-03-26 EP disclosed
WO-2007008895-A1 KINASE INHIBITORS ALLERGAN, INC. (US) 2007-01-18 WO disclosed