SCHEMBL4789757

SCHEMBL4789757

CN1CCC(N(Cc2cccn2C)S(=O)(=O)c2ccc(Nc3ncc(-c4ccc(F)cc4)c(N)n3)cc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.41
PTGS1 P23219 1/20 0.41
HTR2A P28223 3/20 0.38
HTR2C P28335 1/20 0.38
JAK2 O60674 2/20 0.38
JAK3 P52333 2/20 0.38
PTK2 Q05397 2/20 0.38
APOBEC3A P31941 1/20 0.38
APOBEC3G Q9HC16 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
HTR1A P08908 2/20 0.38
DRD2 P14416 2/20 0.38
HTR7 P34969 2/20 0.38
EGFR P00533 2/20 0.37
CDK4 P11802 2/20 0.37
CCND1 P24385 2/20 0.37
CCNT1 O60563 1/20 0.37
CCNE1 P24864 1/20 0.37
CDK2 P24941 1/20 0.37
CDK9 P50750 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4789756 0.90 EGFR (0.40) PTGS2PTGS1HTR2AHTR2CAPOBEC3A
SCHEMBL4884806 0.85 MEN1 (0.43) HTR2AHTR2CJAK2JAK3APOBEC3A
SCHEMBL14020090 0.78 JAK2 (0.41) JAK2JAK3EGFRCDK4CCNE1
SCHEMBL4708985 0.78 AXL (0.41) JAK2CDK4CCND1AXLMAP4K1
SCHEMBL14625275 0.75 HTR2A (0.44) HTR2AHTR2CL3MBTL1MAPT
SCHEMBL4753976 0.74 TNK2 (0.42) JAK2AXL
SCHEMBL4883738 0.71 MEN1 (0.50) HTR2AHTR2CJAK2JAK3APOBEC3A
SCHEMBL4621951 0.71 MEN1 (0.47) HTR2AHTR2CJAK2JAK3APOBEC3A
SCHEMBL4622666 0.71 MEN1 (0.47) HTR2AHTR2CJAK2JAK3APOBEC3A
Hydrochloric Acid SCHEMBL4886318 0.70 MEN1 (0.47) HTR2AHTR2CJAK2JAK3APOBEC3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904479-A2 NOVEL 2,4-DIANILINOPYRIMIDINE DERIVATIVES, THE PREPARATION THEREOF, THEIR USE AS MEDICAMENTS, PHARMACEUTICAL COMPOSITIONS AND, IN PARTICULAR, AS IKK INHIBITORS Sanofi-Aventis (FR) 2008-04-02 EP disclosed
WO-2007006926-A2 NOVEL 2,4-DIANILINOPYRIMIDINE DERIVATIVES, THE PREPARATION THEREOF, THEIR USE AS MEDICAMENTS, PHARMACEUTICAL COMPOSITIONS AND, IN PARTICULAR, AS IKK INHIBITORS SANOFI-AVENTIS (FR) 2007-01-18 WO disclosed