SCHEMBL4789937

SCHEMBL4789937

COc1cc(C2=C(c3ccccc3)C(=O)NC2=O)cc(OC)c1OC

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 16/20 0.67
FLT3 P36888 9/20 0.64
GSK3B P49841 9/20 0.64
PDGFRB P09619 5/20 0.64
IGF1R P08069 4/20 0.64
KIT P10721 4/20 0.64
PDGFRA P16234 4/20 0.64
FLT1 P17948 4/20 0.64
FLT4 P35916 4/20 0.64
TEK Q02763 4/20 0.64
EGFR P00533 3/20 0.64
ERBB2 P04626 3/20 0.64
PLK4 O00444 1/20 0.64
AURKA O14965 1/20 0.64
NUAK1 O60285 1/20 0.64
ABL1 P00519 1/20 0.64
INSR P06213 1/20 0.64
MET P08581 1/20 0.64
CDK4 P11802 1/20 0.64
SRC P12931 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10629414 0.84 KDR (0.52) KDRFLT3GSK3BPDGFRBIGF1R
SCHEMBL27941836 0.84 KDR (0.67) KDRFLT3GSK3BPDGFRBIGF1R
SCHEMBL27983199 0.83 PDE4B (0.52) KDRFLT3GSK3BPDGFRBIGF1R
SCHEMBL1155691 0.83 KDR (0.63) KDRFLT3GSK3BPDGFRBIGF1R
SCHEMBL4752042 0.82 ALDH1A1 (0.54) KDRFLT3GSK3BPDGFRBIGF1R
SCHEMBL1155579 0.80 KDR (0.59) KDRFLT3GSK3BPDGFRBIGF1R
SCHEMBL3823447 0.79 STK10 (0.66) GSK3B
Maleimide SCHEMBL1155440 0.79 KDR (1.00) KDRFLT3GSK3BPDGFRBIGF1R
SCHEMBL1155976 0.78 KDR (0.63) KDRFLT3GSK3BPDGFRBIGF1R
SCHEMBL1155542 0.77 KDR (1.00) KDRFLT3GSK3BPDGFRBFLT4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008140251-A2 CYCLOOXYGENASE-2 INHIBITORS UNIVERSITY-INDUSTRY COOPERATION GROUP OF KYUNG HEE UNIVERSITY (KR) 2008-11-20 WO disclosed