SCHEMBL4790381

SCHEMBL4790381

O=C(O)c1ccc(CN2CC3CC2CN3Cc2ccc(OCC(F)(F)F)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 7/20 0.59
ALDH1A1 P00352 1/20 0.46
PTGER4 P35408 1/20 0.43
NR4A2 P43354 3/20 0.42
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
STAT3 P40763 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40
RXRA P19793 1/20 0.40
HNF4A P41235 1/20 0.40
PDGFRA P16234 1/20 0.40
S1PR1 P21453 1/20 0.40
S1PR5 Q9H228 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3036716 1.00 LTA4H (0.59) LTA4HALDH1A1PTGER4NR4A2CYP2C9
SCHEMBL3041244 0.91 LTA4H (0.57) LTA4HALDH1A1PTGER4NR4A2RXRA
SCHEMBL3040886 0.89 LTA4H (0.55) LTA4HALDH1A1PTGER4NR4A2
SCHEMBL3032148 0.89 LTA4H (0.55) LTA4HALDH1A1PTGER4NR4A2RXRA
SCHEMBL4790531 0.88 LTA4H (0.57) LTA4HPTGER4NR4A2S1PR1S1PR5
SCHEMBL3038132 0.88 LTA4H (0.57) LTA4HPTGER4NR4A2S1PR1S1PR5
SCHEMBL3042632 0.87 LTA4H (0.56) LTA4HS1PR1S1PR5
SCHEMBL3042634 0.87 LTA4H (0.56) LTA4HS1PR1S1PR5
SCHEMBL3041064 0.87 LTA4H (0.53) LTA4HALDH1A1PTGER4NR4A2RXRA
SCHEMBL3036296 0.85 LTA4H (0.56) LTA4HPTGER4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1976828-A1 DIAMINE DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE Schering Aktiengesellschaft (DE) 2008-10-08 EP disclosed
WO-2007079078-A1 DIAMINE DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2007-07-12 WO disclosed