SCHEMBL4792253

SCHEMBL4792253

CNCc1cc(-c2cccc(C(C)OC(=O)/C=C/C(=O)O)c2F)n(S(=O)(=O)c2cccnc2)c1

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.32
MEN1 O00255 1/20 0.31
POLB P06746 1/20 0.31
KMT2A Q03164 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
HSD17B10 Q99714 1/20 0.31
NAMPT P43490 6/20 0.30
KAT5 Q92993 1/20 0.30
KAT8 Q9H7Z6 1/20 0.30
ALDH1A1 P00352 2/20 0.30
HDAC1 Q13547 2/20 0.30
PTGDR2 Q9Y5Y4 1/20 0.30
HDAC3 O15379 1/20 0.30
HDAC4 P56524 1/20 0.30
HDAC7 Q8WUI4 1/20 0.30
HDAC2 Q92769 1/20 0.30
HDAC10 Q969S8 1/20 0.30
HDAC11 Q96DB2 1/20 0.30
HDAC8 Q9BY41 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1278430 0.97 HSD17B10 (0.32) HSD17B10NAMPTALDH1A1HDAC1HDAC3
Fumaric Acid SCHEMBL1278431 0.90 HSD17B10 (0.33) MEN1POLBKMT2AL3MBTL1HSD17B10
Fumaric Acid SCHEMBL1278428 0.90 HSD17B10 (0.33) MEN1POLBKMT2AL3MBTL1HSD17B10
SCHEMBL4793307 0.85 HCAR2 (0.38) HCAR2MEN1POLBKMT2AL3MBTL1
Fumaric Acid SCHEMBL1278492 0.85 NAMPT (0.40) MEN1POLBKMT2AL3MBTL1HSD17B10
Fumaric Acid SCHEMBL1278489 0.85 NAMPT (0.40) MEN1POLBKMT2AL3MBTL1HSD17B10
SCHEMBL1580592 0.84 EPHX2 (0.34) HSD17B10NAMPTKAT5KAT8ALDH1A1
Fumaric Acid SCHEMBL1278703 0.84 KAT8 (0.36) MEN1POLBKMT2AL3MBTL1NAMPT
Fumaric Acid SCHEMBL1278371 0.84 NAMPT (0.35) MEN1POLBKMT2AL3MBTL1NAMPT
Fumaric Acid SCHEMBL1278699 0.84 KAT8 (0.36) MEN1POLBKMT2AL3MBTL1NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919865-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2008-05-14 EP disclosed
WO-2007026916-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-03-08 WO disclosed