SCHEMBL4793307

SCHEMBL4793307

CNCc1cc(-c2cccc(COC(=O)/C=C/C(=O)O)c2F)n(S(=O)(=O)c2cccnc2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 4/20 0.38
EPHX1 P07099 1/20 0.34
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33
MEN1 O00255 1/20 0.33
POLB P06746 1/20 0.33
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KAT5 Q92993 1/20 0.33
KAT8 Q9H7Z6 1/20 0.33
AOC3 Q16853 2/20 0.31
ALDH1A1 P00352 2/20 0.31
NAMPT P43490 2/20 0.31
HDAC1 Q13547 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
TSHR P16473 1/20 0.31
KDM6B O15054 1/20 0.30
ALKBH2 Q6NS38 1/20 0.30
ALKBH3 Q96Q83 1/20 0.30
FTO Q9C0B1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1278370 0.97 EPHX1 (0.35) HCAR2EPHX1PDCD1CD274KAT5
Fumaric Acid SCHEMBL1278367 0.90 NAMPT (0.35) EPHX1PDCD1CD274MEN1POLB
Fumaric Acid SCHEMBL1278371 0.90 NAMPT (0.35) EPHX1PDCD1CD274MEN1POLB
SCHEMBL1278824 0.89 EPHX1 (0.36) EPHX1ALDH1A1NAMPTHDAC1TSHR
Fumaric Acid SCHEMBL1278489 0.86 NAMPT (0.40) MEN1POLBKMT2AL3MBTL1ALDH1A1
Fumaric Acid SCHEMBL1278492 0.86 NAMPT (0.40) MEN1POLBKMT2AL3MBTL1ALDH1A1
Fumaric Acid SCHEMBL1278703 0.85 KAT8 (0.36) MEN1POLBKMT2AL3MBTL1KAT5
Fumaric Acid SCHEMBL1278699 0.85 KAT8 (0.36) MEN1POLBKMT2AL3MBTL1KAT5
SCHEMBL4792253 0.85 HCAR2 (0.32) HCAR2MEN1POLBKMT2AL3MBTL1
Fumaric Acid SCHEMBL1278205 0.85 KAT5 (0.36) MEN1POLBKMT2AL3MBTL1KAT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919865-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2008-05-14 EP disclosed
WO-2007026916-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-03-08 WO disclosed