SCHEMBL4792299

SCHEMBL4792299

CC(C)[C@@H]1C(=O)[C@@H](NC(=O)OC(C)(C)C)C(=O)N1C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 5/20 0.38
NFKB2 Q00653 5/20 0.38
RELA Q04206 5/20 0.38
GAA P10253 1/20 0.35
KMT2A Q03164 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CTSK P43235 2/20 0.32
KLK7 P49862 1/20 0.31
KLK5 Q9Y337 1/20 0.31
BTK Q06187 1/20 0.31
CHRM2 P08172 1/20 0.31
CHRM1 P11229 1/20 0.31
CHRM3 P20309 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA7 P43166 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4790633 0.72 KLK7 (0.34) NFKB1NFKB2RELAL3MBTL1KLK7
SCHEMBL13391275 0.70 NFKB1 (0.42) NFKB1NFKB2RELAGAAKMT2A
SCHEMBL3692487 0.68 NFKB1 (0.32) NFKB1NFKB2RELA
SCHEMBL3302910 0.68 NFKB1 (0.32) NFKB1NFKB2RELA
SCHEMBL14515887 0.68 CHRM2 (0.38) L3MBTL1KLK7KLK5CHRM2CHRM1
SCHEMBL34475689 0.68 CHRM2 (0.38) L3MBTL1KLK7KLK5CHRM2CHRM1
SCHEMBL13391516 0.68 NFKB1 (0.31) NFKB1NFKB2RELA
SCHEMBL2132635 0.67 KLK7 (0.33) L3MBTL1KLK7KLK5CHRM2CHRM1
SCHEMBL2132631 0.67 KLK7 (0.33) L3MBTL1KLK7KLK5CHRM2CHRM1
SCHEMBL4792104 0.67 PLA2G10 (0.36) L3MBTL1KLK7KLK5CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2134681-B1 TRANS-ANNULAR REARRANGEMENT OF ACTIVE LACTAMES CENTRE NAT RECH SCIENT (FR) 2012-05-16 EP disclosed
WO-2008125421-A1 TRANS-ANNULAR REARRANGEMENT OF ACTIVE LACTAMES CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2008-10-23 WO disclosed