SCHEMBL4792597

SCHEMBL4792597

CS(=O)(=O)[As](Cc1cccc(Cl)c1Cl)c1ccc(N(C=O)CC(O)c2ccccc2)cc1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP51A1 Q16850 1/20 0.32
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32
AOC3 Q16853 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
MAPK1 P28482 1/20 0.30
CACNA2D1 P54289 2/20 0.30
CACNA1B Q00975 2/20 0.30
CACNB1 Q02641 2/20 0.30
CACNA1C Q13936 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4777314 0.82 GAA (0.38) NR1H2NR1H3MAPK1
SCHEMBL4777570 0.76 GAA (0.43) CYP51A1NR1H2NR1H3MAPK1
SCHEMBL4777561 0.71 GAA (0.36) MAPK1
SCHEMBL4775362 0.69 GAA (0.39) SLC6A2SLC6A4
SCHEMBL4771365 0.67 GAA (0.37) MAPK1
SCHEMBL4777347 0.67 NR1H4 (0.39) SLC6A2SLC6A4
SCHEMBL4776590 0.63 GAA (0.42) MAPK1
SCHEMBL4767994 0.61 GAA (0.53)
SCHEMBL4775060 0.60 GAA (0.39)
SCHEMBL16155387 0.58 AOC3 (0.59) AOC3SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1942888-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-07-16 EP claimed
WO-2007056078-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-18 WO claimed