SCHEMBL4795265

SCHEMBL4795265

COC(=O)c1nn(-c2ccc(C(F)(F)F)cc2)c2ccc(C)cc12

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.57
ADORA1 P30542 1/20 0.45
ATM Q13315 1/20 0.43
ELANE P08246 4/20 0.43
ALDH1A1 P00352 3/20 0.41
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
F2 P00734 2/20 0.41
PLAU P00749 2/20 0.41
CTRB1 P17538 1/20 0.41
POLB P06746 1/20 0.40
NR3C1 P04150 1/20 0.40
NPY5R Q15761 1/20 0.39
NPBWR1 P48145 1/20 0.39
MCHR1 Q99705 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4790806 0.88 SCN9A (0.72) SCN9AADORA1ATMELANEALDH1A1
SCHEMBL4792382 0.87 SCN9A (0.62) SCN9AATMELANEALDH1A1KMT2A
SCHEMBL4795594 0.87 SCN9A (0.56) SCN9AADORA1ATMALDH1A1KMT2A
SCHEMBL4792532 0.86 SCN9A (0.61) SCN9AADORA1ATMELANEALDH1A1
SCHEMBL4791726 0.84 SCN9A (0.55) SCN9AADORA1ATMELANEF2
SCHEMBL4794092 0.81 SCN9A (0.48) SCN9AADORA1ATMKMT2AMEN1
SCHEMBL4794087 0.78 SCN9A (0.42) SCN9AATMNR3C1NPY5RNPBWR1
SCHEMBL25678102 0.78 SCN9A (0.44) SCN9AATMPOLBNR3C1CYP2C9
SCHEMBL16260376 0.76 SCN9A (0.56) SCN9AELANEALDH1A1KMT2AMEN1
SCHEMBL12070101 0.76 SCN9A (0.74) SCN9AADORA1ELANEALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937647-A1 CONDENSED PYRAZOLE DERIVATIVES AS PPAR AGONISTS II Inpharmatica Limited (GB) 2008-07-02 EP disclosed
WO-2007036727-A1 CONDENSED PYRAZOLE DERIVATIVES AS PPAR AGONISTS II INPHARMATICA LIMITED (GB) 2007-04-05 WO disclosed
WO-2007036727-A1 CONDENSED PYRAZOLE DERIVATIVES AS PPAR AGONISTS II INPHARMATICA LIMITED (GB) 2007-04-05 WO disclosed