SCHEMBL4795825

SCHEMBL4795825

CC(C)C(NCCC[AsH2])c1oc2cc(F)ccc2c(=O)c1Cc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.39
KIF11 P52732 1/20 0.39
HSD17B3 P37058 2/20 0.36
KDM4E B2RXH2 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ERAP1 Q9NZ08 1/20 0.36
ACP1 P24666 4/20 0.36
PTPN1 P18031 2/20 0.36
MCHR1 Q99705 1/20 0.35
ESR1 P03372 1/20 0.35
AR P10275 1/20 0.35
NQO1 P15559 2/20 0.33
MAOB P27338 1/20 0.33
PLA2G2A P14555 1/20 0.33
CYP11B1 P15538 2/20 0.33
CYP11B2 P19099 2/20 0.33
CYP17A1 P05093 1/20 0.32
CYP19A1 P11511 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3270268 0.91 KCNH2 (0.46) KCNH2KIF11HSD17B3KDM4EGLA
SCHEMBL3269493 0.91 KCNH2 (0.46) KCNH2KIF11HSD17B3KDM4EGLA
SCHEMBL12735758 0.81 KCNH2 (0.40) KCNH2KIF11HSD17B3KDM4EGLA
SCHEMBL11920180 0.80 KIF11 (0.51) KCNH2KIF11HSD17B3KDM4EGLA
SCHEMBL3313494 0.80 KCNH2 (0.43) KCNH2KIF11MCHR1MAOB
SCHEMBL3271196 0.79 KIF11 (0.58) KCNH2KIF11HSD17B3KDM4EGLA
SCHEMBL3268480 0.79 KCNH2 (0.37) KCNH2KIF11GLAMCHR1NQO1
SCHEMBL13309014 0.79 KCNH2 (0.44) KCNH2KIF11HSD17B3KDM4EGLA
SCHEMBL10192157 0.77 PPARG (0.47) KCNH2KIF11HSD17B3KDM4EGLA
SCHEMBL3269903 0.77 KIF11 (0.45) KCNH2KIF11HSD17B3KDM4EGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1956908-A2 CERTAIN COMPOSITIONS AND METHODS OF TREATMENT Cytokinetics, Inc. (US) 2008-08-20 EP disclosed
WO-2007067752-A2 CERTAIN COMPOSITIONS AND METHODS OF TREATMENT CYTOKINETICS, INC. (US) 2007-06-14 WO disclosed