SCHEMBL479899

SCHEMBL479899

Cc1cc(C(O)(C(C)c2ccc(Oc3cc(C(F)(F)F)c(C(=O)O)cn3)cc2Cl)C(F)(F)F)c[nH]c1=O

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.35
MAPK10 P53779 7/20 0.35
MAPK8 P45983 3/20 0.35
KDM4E B2RXH2 4/20 0.35
ALDH1A1 P00352 2/20 0.35
NPC1 O15118 1/20 0.35
MAPK1 P28482 1/20 0.35
GABRA5 P31644 1/20 0.34
RAF1 P04049 1/20 0.33
MAPK3 P27361 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
GAA P10253 2/20 0.31
MCOLN3 Q8TDD5 1/20 0.31
KDR P35968 2/20 0.31
BRAF P15056 1/20 0.31
POLB P06746 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL479991 0.92 MAPT (0.45) MAPTMAPK10MAPK8KDM4EALDH1A1
SCHEMBL480052 0.89 RHEB (0.35) MEN1KMT2AKDR
SCHEMBL473801 0.86 MAPT (0.36) MAPTMAPK10MAPK8KDM4EALDH1A1
SCHEMBL12164133 0.86 MAPT (0.36) MAPTMAPK10MAPK8KDM4EALDH1A1
SCHEMBL480607 0.85 MAPT (0.35) MAPTMAPK10MAPK8KDM4EALDH1A1
SCHEMBL753346 0.85 MAPT (0.35) MAPTMAPK10MAPK8KDM4EALDH1A1
SCHEMBL479931 0.85 S1PR2 (0.33) MEN1KMT2A
SCHEMBL732783 0.83 MAPK10 (0.37) MAPTMAPK10MAPK8KDM4EALDH1A1
SCHEMBL752281 0.83 MAPK10 (0.37) MAPTMAPK10MAPK8KDM4EALDH1A1
SCHEMBL755682 0.83 MAPT (0.35) MAPTMAPK10MAPK8KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP claimed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO claimed
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed