SCHEMBL480052

SCHEMBL480052

Cc1cc(C(O)(C(C)c2ccc(Oc3ccc(C(=O)O)c(C(F)(F)F)c3)cc2Cl)C(F)(F)F)c[nH]c1=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RHEB Q15382 1/20 0.35
THRA P10827 4/20 0.33
THRB P10828 4/20 0.33
PPARG P37231 4/20 0.32
PPARA Q07869 3/20 0.32
MEN1 O00255 1/20 0.31
TTR P02766 1/20 0.31
PPOX P50336 1/20 0.31
KMT2A Q03164 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
KDR P35968 2/20 0.31
FLT1 P17948 1/20 0.31
PPARD Q03181 2/20 0.30
MRGPRX4 Q96LA9 1/20 0.30
PRKAB2 O43741 1/20 0.30
PRKAG1 P54619 1/20 0.30
PRKAA2 P54646 1/20 0.30
PRKAA1 Q13131 1/20 0.30
PRKAG3 Q9UGI9 1/20 0.30
PRKAG2 Q9UGJ0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL479931 0.94 S1PR2 (0.33) THRATHRBPPARGPPARAMEN1
SCHEMBL480020 0.91 PRKAB2 (0.33) PPARGPPARAPPARDPRKAB2PRKAG1
SCHEMBL479899 0.89 MAPT (0.35) MEN1KMT2AKDR
SCHEMBL480101 0.89 MCL1 (0.35) THRATHRBKDRFLT1CHEK2
SCHEMBL480000 0.88 S1PR2 (0.33) THRATHRBPPARGPPARAMEN1
SCHEMBL479964 0.87 KDR (0.32) THRATHRBPPARGPPARAKMT2A
SCHEMBL480031 0.85 KMT2A (0.32) THRATHRBMEN1TTRPPOX
SCHEMBL479915 0.84 PRKAB2 (0.33) THRATHRBPPARGPPARAMEN1
SCHEMBL479852 0.84 SMN1; SMN2 (0.40) THRATHRBPPARGPPARAPPARD
SCHEMBL479958 0.84 MCL1 (0.41) THRATHRBPPARGPPARAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP claimed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO claimed
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed