SCHEMBL4803018

SCHEMBL4803018

O=S(=O)(Cc1cc2ccccc2s1)c1cc2ccccc2s1

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.57
CYP2A6 P11509 4/20 0.51
ASIC3 Q9UHC3 1/20 0.51
LOXL2 Q9Y4K0 1/20 0.51
AGXT P21549 1/20 0.47
ADRB2 P07550 1/20 0.47
AKR1B1 P15121 1/20 0.43
CTRC Q99895 2/20 0.40
ADRA1D P25100 2/20 0.40
CCR2 P41597 1/20 0.40
TPSAB1 Q15661 1/20 0.39
IDH1 O75874 1/20 0.39
CA1 P00915 1/20 0.39
CA9 Q16790 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1272861 0.79 CYP2A6 (0.55) CA2CYP2A6ASIC3LOXL2AGXT
SCHEMBL1272859 0.79 CYP2A6 (0.55) CA2CYP2A6ASIC3LOXL2AGXT
SCHEMBL329294 0.76 CA2 (0.71) CA2CYP2A6ASIC3LOXL2AKR1B1
SCHEMBL19551366 0.75 CYP2A6 (0.50) CA2CYP2A6ASIC3LOXL2AGXT
SCHEMBL1416155 0.75 CA2 (0.65) CA2CYP2A6ASIC3LOXL2AKR1B1
SCHEMBL329449 0.74 CA2 (0.69) CA2CYP2A6ASIC3LOXL2AKR1B1
SCHEMBL9350079 0.74 CA2 (0.54) CA2CYP2A6ASIC3LOXL2AGXT
SCHEMBL25119616 0.73 CA2 (0.67) CA2CYP2A6ASIC3LOXL2AKR1B1
SCHEMBL743918 0.73 CA2 (0.67) CA2CYP2A6ASIC3LOXL2AKR1B1
SCHEMBL792780 0.73 CA2 (1.00) CA2CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7381728-B2 Piperazine derivatives useful for the treatment of gastrointestinal disorders GLAXO GROUP LIMITED (GB) 2008-06-03 US disclosed