SCHEMBL4803305

SCHEMBL4803305

C1=CN(Nc2ccccc2)CN=C1

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.32
TDP1 Q9NUW8 2/20 0.32
ALDH1A1 P00352 1/20 0.30
CTSD P07339 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3681186 0.69 TDP1 (0.37) CYP1A2TDP1ALDH1A1CTSDHSD17B10
SCHEMBL1226360 0.68 CYP2C9 (0.43) ALDH1A1
SCHEMBL10883415 0.67
SCHEMBL2362320 0.67 MAPT (0.35) ALDH1A1
SCHEMBL7453603 0.65
SCHEMBL10864613 0.65 CYP1A2 (0.34) CYP1A2TDP1ALDH1A1CTSDHSD17B10
SCHEMBL1036360 0.65 LMNA (0.34) CYP1A2TDP1ALDH1A1CTSDHSD17B10
Hydrochloric Acid SCHEMBL27419243 0.64 POLB (0.34) CYP1A2TDP1ALDH1A1CTSDHSD17B10
SCHEMBL4803312 0.63 TDP1 (0.35) CYP1A2TDP1ALDH1A1CTSDHSD17B10
SCHEMBL1413144 0.63

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101511800-B Triazolyl phenyl benzenesulfonamides CHEMOCENTRYX INC 2013-02-27 CN disclosed
CN-101511800-A Triazolyl phenyl benzenesulfonamides CHEMOCENTRYX INC (US) 2009-08-19 CN disclosed
US-7329661-B2 N-phenyl-3-pyrimidine-amine derivatives NOVARTIS AG (CH) 2008-02-12 US disclosed