SCHEMBL4804728

SCHEMBL4804728

O=C(OCc1ccccc1)N(Cc1ccccc1)C1CCC(OCCCCCCN2CCOCC2)CC1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BCHE P06276 11/20 0.48
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
ACHE P22303 1/20 0.43
ABCB1 P08183 1/20 0.43
OPRM1 P35372 1/20 0.42
TRPV4 Q9HBA0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4804735 1.00 BCHE (0.48) BCHEALDH1A1KDM4ESMN1; SMN2TDP1
SCHEMBL4802417 0.93 BCHE (0.48) BCHEALDH1A1KDM4ESMN1; SMN2TDP1
SCHEMBL4802422 0.93 BCHE (0.48) BCHEALDH1A1KDM4ESMN1; SMN2TDP1
SCHEMBL4804719 0.92 BCHE (0.51) BCHEALDH1A1KDM4ESMN1; SMN2ACHE
SCHEMBL4804843 0.92 BCHE (0.51) BCHEALDH1A1KDM4EACHEOPRM1
SCHEMBL4804836 0.92 BCHE (0.51) BCHEALDH1A1KDM4EACHEOPRM1
SCHEMBL4804726 0.92 BCHE (0.51) BCHEALDH1A1KDM4ESMN1; SMN2ACHE
SCHEMBL4805112 0.90 CCR5 (0.48) BCHE
SCHEMBL4805101 0.90 CCR5 (0.48) BCHE
SCHEMBL4806551 0.89 HTR2A (0.49) BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1311475-B1 AMINOCYCLOHEXANE DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-08-06 EP disclosed
US-7335687-B2 2,3-Oxidosqualene-lanosterol cyclase inhibitors HOFFMANN-LA ROCHE INC. (US) 2008-02-26 US disclosed
US-20050176766-A1 2,3-Oxidosqualene-lanosterol cyclase inhibitors ACKERMANN JEAN (CH) 2005-08-11 US disclosed
US-6858651-B2 2,3-oxidosqualene-lanosterol cyclase inhibitors HOFFMANN-LA ROCHE INC. (US) 2005-02-22 US disclosed
CN-1468214-A Novel derivatives of aminocyclohexane - 2004-01-14 CN disclosed
EP-1311475-A1 NOVEL AMINOCYCLOHEXANE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2003-05-21 EP disclosed
US-20020045777-A1 2,3-oxidosqualene-lanosterol cyclase inhibitors F.HOFFMANN-LA ROCHE AG (CH) 2002-04-18 US disclosed
WO-2002014267-A1 NOVEL AMINOCYCLOHEXANE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-02-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050176766-A1 2,3-Oxidosqualene-lanosterol cyclase inhibitors CYP51A1, LSS, CYP46A1 BCHE 736/4885ALDH1A1 2260/4885KDM4E 4198/4885
US-20020045777-A1 2,3-oxidosqualene-lanosterol cyclase inhibitors CYP51A1, LSS, CYP46A1 BCHE 736/4885ALDH1A1 2260/4885KDM4E 4198/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.