SCHEMBL4805555

SCHEMBL4805555

CNS(=O)(=O)Oc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.55
MEN1 O00255 2/20 0.55
CA2 P00918 5/20 0.52
CA1 P00915 3/20 0.52
CA9 Q16790 3/20 0.52
PPARG P37231 4/20 0.47
NFE2L2 Q16236 2/20 0.47
LMNA P02545 1/20 0.47
CA12 O43570 1/20 0.45
SLC40A1 Q9NP59 1/20 0.42
PGR P06401 1/20 0.41
ALDH1A1 P00352 1/20 0.39
CA4 P22748 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
HPGD P15428 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27699140 0.98 KMT2A (0.53) KMT2AMEN1CA2CA1CA9
SCHEMBL27545486 0.88 CA2 (0.59) KMT2AMEN1CA2CA1CA9
SCHEMBL9365762 0.80 CA2 (0.57) KMT2AMEN1CA2CA1CA9
SCHEMBL9451309 0.78 CA2 (0.55) KMT2AMEN1CA2CA1CA9
SCHEMBL323791 0.78 CA1 (0.58) KMT2AMEN1CA2CA1CA9
SCHEMBL10736241 0.77 KMT2A (0.60) KMT2AMEN1CA2CA1CA9
SCHEMBL20768536 0.77 KMT2A (0.60) KMT2AMEN1CA2CA1CA9
SCHEMBL29171358 0.77 KMT2A (0.55) KMT2AMEN1CA2CA1CA9
SCHEMBL27390987 0.77 KMT2A (0.55) KMT2AMEN1CA2CA1CA9
SCHEMBL9451377 0.77 KMT2A (0.50) KMT2AMEN1CA2CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5025031-A Aryl and aryloxyalkyl sulfamate esters useful as anticonvulsants A. H. ROBINS CO., INC. (US) 1991-06-18 US claimed
EP-0403185-A2 Compounds having one or more aminosulfonyloxy radicals useful as pharmaceuticals A.H. ROBINS COMPANY, INCORPORATED (US) 1990-12-19 EP claimed
CN-104725856-B Conductive composition and the electric conductor and solid electrolytic capacitor of above-mentioned conductive composition are used 三菱丽阳株式会社 2017-06-09 CN disclosed
US-7335687-B2 2,3-Oxidosqualene-lanosterol cyclase inhibitors HOFFMANN-LA ROCHE INC. (US) 2008-02-26 US disclosed
US-20050176766-A1 2,3-Oxidosqualene-lanosterol cyclase inhibitors ACKERMANN JEAN (CH) 2005-08-11 US disclosed
US-6858651-B2 2,3-oxidosqualene-lanosterol cyclase inhibitors HOFFMANN-LA ROCHE INC. (US) 2005-02-22 US disclosed
CN-1119457-C Method for improving wet strength of paper KIMBERLY CLARK CO (US) 2003-08-27 CN disclosed
CN-1341571-A Aminosulfonic acid series high-effective water-reducing agent and its preparation method HUA NAN UNIVERSITY OF SCIENCE (CN) 2002-03-27 CN disclosed
CN-1292838-A Method for improving wet strength of paper KIMBERLY CLARK CO (US) 2001-04-25 CN disclosed
US-5273993-A Antiarthritic agents; osteoporosis A. H. ROBINS COMPANY, INCORPORATED (US) 1993-12-28 US disclosed
US-5194446-A Antiarthritic agents A. H. ROBINS COMPANY, INCORPORATED (US) 1993-03-16 US disclosed
US-5192785-A Sulfamates as antiglaucoma agents A. H. ROBINS COMPANY, INCORPORATED (US) 1993-03-09 US disclosed
US-5025031-A Aryl and aryloxyalkyl sulfamate esters useful as anticonvulsants A. H. ROBINS CO., INC. (US) 1991-06-18 US disclosed
EP-0403185-A2 Compounds having one or more aminosulfonyloxy radicals useful as pharmaceuticals A.H. ROBINS COMPANY, INCORPORATED (US) 1990-12-19 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050176766-A1 2,3-Oxidosqualene-lanosterol cyclase inhibitors CYP51A1, LSS, CYP46A1 KMT2A 3998/4885MEN1 429/4885CA2 2022/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.