SCHEMBL480695

SCHEMBL480695

CN(c1ccc(S(=O)(=O)O)cc1)c1ccccc1-c1cnc2nc(N)nc(N)c2n1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CA1 P00915 6/20 0.48
CA2 P00918 6/20 0.48
PIK3CG P48736 3/20 0.41
DHFR P00374 8/20 0.41
PIK3CA P42336 1/20 0.41
PIK3CB P42338 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
CA9 Q16790 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13583145 0.81 CA1 (0.55) CA1CA2PIK3CGDHFRCA9
SCHEMBL480692 0.72 CA1 (0.61) CA1CA2DHFRCA9
SCHEMBL8813941 0.70 PIK3CG (0.54) PIK3CGDHFRPIK3CAPIK3CBHDAC6
SCHEMBL3755689 0.65 NOS1 (0.42) DHFR
SCHEMBL13187327 0.65 CA1 (1.00) CA1CA2DHFRCA9
SCHEMBL8813951 0.65 PIK3CG (0.72) PIK3CGDHFRPIK3CAPIK3CBHDAC6
SCHEMBL3761058 0.64 PIK3CG (0.53) PIK3CGDHFRPIK3CAPIK3CBHDAC6
SCHEMBL479287 0.63 HDAC4 (0.48) CA1CA2PIK3CGDHFRCA9
SCHEMBL3763640 0.63 NOS1 (0.68) PIK3CGPIK3CA
SCHEMBL4130539 0.62 TSHR (0.58) CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2410856-A1 DIAMINOPTERIDINE DERIVATIVES Biorelix, Inc. (US) 2012-02-01 EP disclosed
WO-2010110907-A1 DIAMINOPTERIDINE DERIVATIVES BIORELIX, INC. (US) 2010-09-30 WO disclosed