SCHEMBL4808925

SCHEMBL4808925

CC(C)(C)C1=CC[CH]C(c2ccc3ccccc3c2)=C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSTP1 P09211 1/20 0.35
ESR1 P03372 1/20 0.35
ESR2 Q92731 1/20 0.35
ALOX5 P09917 1/20 0.34
CA1 P00915 2/20 0.33
CA9 Q16790 2/20 0.33
HSD17B1 P14061 1/20 0.33
HSD17B2 P37059 1/20 0.33
CA12 O43570 1/20 0.33
NISCH Q9Y2I1 1/20 0.33
ABL1 P00519 1/20 0.32
SRC P12931 1/20 0.32
CYP1A2 P05177 3/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27459545 0.80 GSTP1 (0.47) GSTP1ESR1ESR2ALOX5CA1
SCHEMBL4004153 0.76 CYP2A6 (0.38) GSTP1ESR1ESR2ALOX5CA1
SCHEMBL4005351 0.76 HTR1D (0.36) GSTP1ESR1ESR2ALOX5CA1
SCHEMBL5887567 0.74 CA1 (0.39) GSTP1ESR1ESR2ALOX5CA1
SCHEMBL5887031 0.74 CDC25A (0.44) GSTP1ESR1ESR2ALOX5CYP1A2
SCHEMBL4009020 0.73 GSTP1 (0.35) GSTP1ESR1ESR2ALOX5HSD17B1
SCHEMBL6897810 0.70 CYP1A2 (0.41) GSTP1ESR1ESR2ALOX5CA1
SCHEMBL21101809 0.66 ESR1 (0.48) GSTP1ESR1ESR2ALOX5CA1
SCHEMBL24795579 0.64 CYP1A2 (0.53) GSTP1ESR1ESR2CA12CYP1A2
SCHEMBL24060806 0.64 GSTP1 (0.41) GSTP1ESR1ESR2ALOX5CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7037931-B2 Corticotropin releasing factor moderator; analgesics; drug abruse, drug dependency; schizophrenia JANSSEN PHARMACEUTICA N.V. (BE) 2006-05-02 US claimed
US-7465808-B2 CCK-1 receptor modulators JANSSEN PHARMACEUTICA, N.V. (BE) 2008-12-16 US disclosed
US-7037931-B2 Corticotropin releasing factor moderator; analgesics; drug abruse, drug dependency; schizophrenia JANSSEN PHARMACEUTICA N.V. (BE) 2006-05-02 US disclosed
US-20060014817-A1 CCK-1 receptor modulators JANSSEN PHARMACEUTICA, N.V. (BE) 2006-01-19 US disclosed
US-20060004195-A1 Alpha,beta-unsaturated esters and acids by stereoselective dehydration JANSSEN PHARMACEUTICA N.V. (BE) 2006-01-05 US disclosed
US-20050026903-A1 CCK-1 receptor modulators JANSSEN PHARMACEUTICA N.V. (BE) 2005-02-03 US disclosed
US-20050020565-A1 Pyrazole compound; gastrointestinal disorders; central nervous system disorders JONES TODD K (US) 2005-01-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050020565-A1 Pyrazole compound; gastrointestinal disorders; central nervous system disorders CCKAR, CCKBR, NPY1R GSTP1 4210/4885ESR1 850/4885ESR2 720/4885
US-20060014817-A1 CCK-1 receptor modulators CCKAR, CCKBR, GIPR GSTP1 4028/4885ESR1 428/4885ESR2 336/4885
US-20060004195-A1 Alpha,beta-unsaturated esters and acids by stereoselective dehydration CCKAR, CCKBR, FFAR1 GSTP1 4217/4885ESR1 207/4885ESR2 122/4885
US-20050026903-A1 CCK-1 receptor modulators CCKAR, CCKBR, GLP1R GSTP1 4526/4885ESR1 202/4885ESR2 176/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.