SCHEMBL4809142

SCHEMBL4809142

Cc1nc(S(C)(=O)=O)nc(C)c1C(=O)N1CC2CN(c3cccc(CCC(N)=O)c3)CC2C1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 16/20 0.41
HCRTR2 O43614 16/20 0.41
USP2 O75604 1/20 0.36
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
KCNH2 Q12809 1/20 0.36
CCL5 P13501 1/20 0.36
PLA2G10 O15496 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4696224 0.89 HCRTR1 (0.39) HCRTR1HCRTR2KCNH2CCL5PLA2G10
SCHEMBL4698184 0.87 HCRTR1 (0.46) HCRTR1HCRTR2
SCHEMBL4968486 0.87 HCRTR1 (0.42) HCRTR1HCRTR2KCNH2CCL5
SCHEMBL5234333 0.86 HCRTR1 (0.41) HCRTR1HCRTR2
SCHEMBL4696692 0.85 HCRTR1 (0.42) HCRTR1HCRTR2KCNH2
SCHEMBL5236658 0.85 HCRTR1 (0.40) HCRTR1HCRTR2KCNH2
SCHEMBL4698030 0.84 HCRTR1 (0.39) HCRTR1HCRTR2KCNH2
SCHEMBL4696182 0.84 HCRTR1 (0.38) HCRTR1HCRTR2KCNH2
SCHEMBL4696183 0.84 HCRTR1 (0.38) HCRTR1HCRTR2KCNH2
SCHEMBL4692413 0.84 HCRTR1 (0.53) HCRTR1HCRTR2KCNH2PLA2G10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed