SCHEMBL4819447

SCHEMBL4819447

COc1ccc(Br)c(C(=O)N2CCN(C(N)C=O)CC2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.53
MAPK1 P28482 1/20 0.53
CPS1 P31327 3/20 0.48
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
PKM P14618 1/20 0.47
CYP2C19 P33261 1/20 0.47
ALDH1A1 P00352 4/20 0.44
MAPT P10636 2/20 0.44
HTT P42858 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
GPR6 P46095 1/20 0.42
HPGD P15428 2/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
DRD3 P35462 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4755205 0.99 KMT2A (0.53) KMT2AMAPK1CPS1CYP1A2CYP3A4
SCHEMBL3759104 0.79 KMT2A (0.55) KMT2AMAPK1CPS1CYP1A2CYP3A4
SCHEMBL1221923 0.78 KMT2A (0.54) KMT2AMAPK1CPS1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL1221532 0.77 KMT2A (0.53) KMT2AMAPK1CPS1CYP1A2CYP3A4
SCHEMBL1515866 0.76 KMT2A (0.55) KMT2AMAPK1CPS1CYP1A2CYP3A4
SCHEMBL1516226 0.75 KMT2A (0.53) KMT2AMAPK1CPS1ALDH1A1MAPT
SCHEMBL13983665 0.74 KMT2A (0.53) KMT2AMAPK1CPS1CYP1A2CYP3A4
SCHEMBL12894668 0.73 KMT2A (0.52) KMT2AMAPK1CPS1CYP1A2CYP3A4
SCHEMBL31350942 0.70 SMN1; SMN2 (0.57) KMT2AMAPK1CYP3A4ALDH1A1MAPT
SCHEMBL1515934 0.70 PKM (0.59) KMT2AMAPK1PKMALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008157844-A1 NOVEL PIPERAZINE DERIVATIVES AS INHIBITORS OF STEAROYL-COA DESATURASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2008-12-24 WO disclosed