SCHEMBL4822008

SCHEMBL4822008

O=C1NC(=O)c2ccc(Br)cc2/C1=C/Nc1cc[c]c(C(=O)O)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNB2 O95067 4/20 0.38
CDK1 P06493 4/20 0.38
CCNB1 P14635 4/20 0.38
CCNB3 Q8WWL7 4/20 0.38
HSP90AA1 P07900 3/20 0.38
CCR6 P51684 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CDK4 P11802 1/20 0.36
CCND1 P24385 1/20 0.36
CDK2 P24941 1/20 0.36
MAOA P21397 3/20 0.34
MAOB P27338 3/20 0.34
RAB9A P51151 1/20 0.34
PIM1 P11309 1/20 0.33
PIM3 Q86V86 1/20 0.33
PIM2 Q9P1W9 1/20 0.33
TGM2 P21980 2/20 0.33
MAP1LC3B Q9GZQ8 1/20 0.33
ALDH1A1 P00352 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3561989 0.79 KDM4C (0.46) CCNB2CDK1CCNB1CCNB3HSP90AA1
SCHEMBL3561986 0.79 KDM4C (0.46) CCNB2CDK1CCNB1CCNB3HSP90AA1
SCHEMBL3573963 0.74 KMT2A (0.40) CCNB2CDK1CCNB1CCNB3HSP90AA1
SCHEMBL3573960 0.74 KMT2A (0.40) CCNB2CDK1CCNB1CCNB3HSP90AA1
SCHEMBL3568888 0.71 KMT2A (0.42) CCNB2CDK1CCNB1CCNB3HSP90AA1
SCHEMBL3568884 0.71 KMT2A (0.42) CCNB2CDK1CCNB1CCNB3HSP90AA1
SCHEMBL3573272 0.71 PDGFRB (0.42) CCNB2CDK1CCNB1CCNB3HSP90AA1
SCHEMBL3573276 0.71 PDGFRB (0.42) CCNB2CDK1CCNB1CCNB3HSP90AA1
SCHEMBL3564130 0.70 MAOA (0.40) CCNB2CDK1CCNB1CCNB3HSP90AA1
SCHEMBL3564133 0.70 MAOA (0.40) CCNB2CDK1CCNB1CCNB3HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963273-A2 SUBSTITUTED ISOQUINOLINE-1,3(2H,4H)-DIONES, 1-THIOXO-1,4-DIHYDRO-2H-ISOQUINOLINE-3-ONES AND 1,4-DIHYDRO-3(2H)-ISOQUINOLONES AND USE THEREOF AS KINASE INHIBITORS Wyeth a Corporation of the State of Delaware (US) 2008-09-03 EP disclosed
WO-2007075783-A2 SUBSTITUTED ISOQUINOLINE-1,3(2H,4H)-DIONES, 1-THIOXO-1,4-DIHYDRO-2H-ISOQUINOLINE-3-ONES AND 1,4-DIHYDRO-3(2H)-ISOQUINOLONES AND USE THEREOF AS KINASE INHIBITOR WYETH (US) 2007-07-05 WO disclosed