SCHEMBL4827658

SCHEMBL4827658

CN[C@@H]1CCCN(c2cnc(Br)c(Cl)c2)C1

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.52
CHRNA4 P43681 2/20 0.52
HRH4 Q9H3N8 16/20 0.47
CHRNB4 P30926 1/20 0.47
CHRNA3 P32297 1/20 0.47
DOT1L Q8TEK3 1/20 0.41
SUV39H2 Q9H5I1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4822000 1.00 CHRNB2 (0.52) CHRNB2CHRNA4HRH4CHRNB4CHRNA3
SCHEMBL4827293 0.87 CHRNB2 (0.51) CHRNB2CHRNA4HRH4CHRNB4CHRNA3
SCHEMBL4827854 0.87 CHRNB2 (0.51) CHRNB2CHRNA4HRH4CHRNB4CHRNA3
SCHEMBL4821233 0.85 CHRNB2 (0.52) CHRNB2CHRNA4HRH4DOT1L
SCHEMBL4823942 0.85 CHRNB2 (0.52) CHRNB2CHRNA4HRH4DOT1L
SCHEMBL4826774 0.85 HRH4 (0.47) HRH4DOT1L
SCHEMBL4819954 0.85 HRH4 (0.47) HRH4DOT1L
SCHEMBL4826729 0.81 CHRNB2 (0.58) CHRNB2CHRNA4HRH4CHRNB4CHRNA3
SCHEMBL4820627 0.81 CHRNB2 (0.58) CHRNB2CHRNA4HRH4CHRNB4CHRNA3
SCHEMBL4826171 0.81 CHRNB2 (0.54) CHRNB2CHRNA4HRH4CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7332504-B2 Heterocyclic substituted aminoazacycles useful as central nervous system agents ABBOTT LABORATORIES (US) 2008-02-19 US claimed
US-7332504-B2 Heterocyclic substituted aminoazacycles useful as central nervous system agents ABBOTT LABORATORIES (US) 2008-02-19 US disclosed