SCHEMBL4827892

SCHEMBL4827892

N[C@@H]1CCCN(c2cnc(Br)c(F)c2)C1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 2/20 0.42
EIF2AK4 Q9P2K8 1/20 0.41
CHRNB2 P17787 6/20 0.40
CHRNA4 P43681 6/20 0.40
CHRNB4 P30926 5/20 0.40
CHRNA3 P32297 5/20 0.40
DPP4 P27487 4/20 0.39
HRH4 Q9H3N8 2/20 0.39
DOT1L Q8TEK3 1/20 0.38
PBK Q96KB5 1/20 0.37
PIM3 Q86V86 1/20 0.37
PIM2 Q9P1W9 1/20 0.37
MAP4K4 O95819 2/20 0.36
AKT1 P31749 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4828915 1.00 PIM1 (0.42) PIM1EIF2AK4CHRNB2CHRNA4CHRNB4
SCHEMBL4820640 0.83 EIF2AK4 (0.46) PIM1EIF2AK4CHRNB2CHRNA4CHRNB4
SCHEMBL29990018 0.83 PIM1 (0.42) PIM1EIF2AK4DPP4HRH4DOT1L
SCHEMBL4828737 0.83 CHRNB2 (0.56) PIM1EIF2AK4CHRNB2CHRNA4CHRNB4
SCHEMBL4827828 0.83 CHRNB2 (0.56) PIM1EIF2AK4CHRNB2CHRNA4CHRNB4
SCHEMBL23497910 0.83 PIM1 (0.42) PIM1EIF2AK4DPP4HRH4DOT1L
SCHEMBL4826774 0.80 HRH4 (0.47) HRH4DOT1L
SCHEMBL4819954 0.80 HRH4 (0.47) HRH4DOT1L
SCHEMBL4827873 0.78 CHRNB2 (0.60) PIM1CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL4827625 0.78 CHRNB2 (0.60) PIM1CHRNB2CHRNA4CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7332504-B2 Heterocyclic substituted aminoazacycles useful as central nervous system agents ABBOTT LABORATORIES (US) 2008-02-19 US claimed
US-7332504-B2 Heterocyclic substituted aminoazacycles useful as central nervous system agents ABBOTT LABORATORIES (US) 2008-02-19 US disclosed