SCHEMBL482835

SCHEMBL482835

CC(=O)N1c2ccc3oc(=O)cc(Cc4ccccc4)c3c2[C@H](OC(N)=O)C[C@@H]1C

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.38
TSHR P16473 1/20 0.38
BRD4 O60885 8/20 0.36
BRD2 P25440 7/20 0.36
BRD3 Q15059 7/20 0.36
HSD17B3 P37058 1/20 0.36
LMNA P02545 3/20 0.36
NPSR1 Q6W5P4 3/20 0.35
MAPT P10636 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL482403 0.86 BRD4 (0.41) BRD4BRD2BRD3HSD17B3
SCHEMBL482791 0.80 HSD17B3 (0.38) TSHRHSD17B3MEN1KMT2AALDH1A1
SCHEMBL482790 0.72 PTGDR2 (0.39) TSHRBRD4MEN1KMT2AALDH1A1
SCHEMBL482474 0.69 SMN1; SMN2 (0.45) SMN1; SMN2TSHRBRD4BRD2BRD3
SCHEMBL482834 0.67 BRD4 (0.30) BRD4LMNAMAPTKDM4EALDH1A1
SCHEMBL482339 0.66 BRD4 (0.40) SMN1; SMN2TSHRBRD4BRD2BRD3
SCHEMBL482769 0.63 NSD2 (0.41) SMN1; SMN2TSHRBRD4
SCHEMBL12095226 0.62 BRD4 (0.51) SMN1; SMN2TSHRBRD4BRD2BRD3
SCHEMBL12095227 0.62 BRD4 (0.51) SMN1; SMN2TSHRBRD4BRD2BRD3
SCHEMBL12095224 0.62 BRD4 (0.51) SMN1; SMN2TSHRBRD4BRD2BRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8604030-B2 Fused piperidine compound and pharmaceutical containing same KOWA COMPANY, LTD. (JP) 2013-12-10 US disclosed
US-20120108581-A1 FUSED PIPERIDINE COMPOUND AND PHARMACEUTICAL CONTAINING SAME KOWA COMPANY, LTD (JP) 2012-05-03 US disclosed
EP-2412710-A1 FUSED PIPERIDINE COMPOUND AND PHARMACEUTICAL AGENT COMPRISING SAME Kowa Company, Ltd. (JP) 2012-02-01 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120108581-A1 FUSED PIPERIDINE COMPOUND AND PHARMACEUTICAL CONTAINING SAME EPOR, JAK2, HBZ SMN1; SMN2 1440/4885TSHR 964/4885BRD4 1271/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.