SCHEMBL4828457

SCHEMBL4828457

CCCCN1C(=O)[C@@H](CC2(O)CCCCC2)NC(=O)C12CCNCC2

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 20/20 0.44
CYP3A4 P08684 2/20 0.42
CYP2C9 P11712 2/20 0.42
CXCR4 P61073 1/20 0.41
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6189687 0.99 CCR5 (0.45) CCR5CYP3A4CYP2C9CXCR4CYP2D6
SCHEMBL5612301 0.89 CCR5 (0.48) CCR5CYP3A4CYP2C9CXCR4CYP2D6
SCHEMBL4828471 0.82 CCR5 (0.44) CCR5CYP3A4CYP2C9CYP2D6
Hydrochloric Acid SCHEMBL5346530 0.82 CCR5 (0.40) CCR5CYP3A4CYP2C9CYP2D6
Hydrochloric Acid SCHEMBL5340685 0.82 CCR5 (0.40) CCR5CYP3A4CYP2C9CYP2D6
SCHEMBL5612320 0.82 CCR5 (0.61) CCR5CYP3A4CYP2C9CYP2D6
SCHEMBL14381400 0.82 CCR5 (0.61) CCR5CYP3A4CYP2C9CYP2D6
SCHEMBL6012736 0.82 CCR5 (0.61) CCR5CYP3A4CYP2C9CYP2D6
Hydrochloric Acid SCHEMBL6186871 0.81 CCR5 (0.56) CCR5CYP3A4CYP2C9CYP2D6
Hydrochloric Acid SCHEMBL5344130 0.81 CCR5 (0.62) CCR5CYP3A4CYP2C9CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7361758-B2 Crystals of triazaspiro[5.5]undecane derivative ONO PHARMACEUTICAL CO., LTD. (JP) 2008-04-22 US disclosed
US-20060052407-A1 Novel crystals of triazaspiro [5.5] undecane derivative ONO PHARMACEUTICAL CO,., LTD (JP) 2006-03-09 US disclosed
EP-1541573-A1 NOVEL CRYSTALS OF TRIAZASPIRO 5.5 UNDECANE DERIVATIVE ONO PHARMACEUTICAL CO., LTD. (JP) 2005-06-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060052407-A1 Novel crystals of triazaspiro [5.5] undecane derivative ACKR3, CCR10, CCR9 CCR5 4/4885CYP3A4 1510/4885CYP2C9 836/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.