SCHEMBL4829599

SCHEMBL4829599

O=C(NC(Cc1ccc(-c2ccc(F)c(Cl)c2)cc1)C(=O)O)c1cc2ccccc2cc1O

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ERAP1 Q9NZ08 2/20 0.51
ECE1 P42892 2/20 0.51
ITGB1 P05556 5/20 0.50
ITGA4 P13612 5/20 0.50
ITGB7 P26010 3/20 0.50
PYGL P06737 1/20 0.49
MME P08473 1/20 0.47
ACE P12821 1/20 0.47
CPA1 P15085 1/20 0.47
ACE2 Q9BYF1 1/20 0.47
GPR34 Q9UPC5 3/20 0.46
HPGDS O60760 1/20 0.45
KIFC1 Q9BW19 1/20 0.45
PDK1 Q15118 1/20 0.45
PDK2 Q15119 1/20 0.45
PDK3 Q15120 1/20 0.45
PDK4 Q16654 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4829604 1.00 ERAP1 (0.51) ERAP1ECE1ITGB1ITGA4ITGB7
SCHEMBL4827784 0.91 ECE1 (0.53) ERAP1ECE1ITGB1ITGA4ITGB7
SCHEMBL4827782 0.91 ECE1 (0.53) ERAP1ECE1ITGB1ITGA4ITGB7
SCHEMBL4824673 0.89 KDR (0.51) ECE1PYGL
SCHEMBL4824679 0.89 KDR (0.51) ECE1PYGL
SCHEMBL27611059 0.88 MME (0.57) ITGB1ITGA4ITGB7MMEACE
SCHEMBL5926558 0.88 MME (0.57) ITGB1ITGA4ITGB7MMEACE
SCHEMBL4827714 0.87 MME (0.47) ERAP1ITGB1ITGA4ITGB7MME
SCHEMBL5927314 0.86 PYGL (0.53) ERAP1ECE1ITGB1ITGA4PYGL
SCHEMBL6497428 0.85 ECE1 (0.52) ERAP1ECE1ITGB1ITGA4ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7459472-B2 Aryl and heteroaryl compounds, compositions, and methods of use TRANSTECH PHARMA, INC. (US) 2008-12-02 US disclosed