SCHEMBL4830639

SCHEMBL4830639

CC(C)(CCn1cnc2nc(OC(=O)O)ccc21)NCC(OC(=O)C(F)(F)F)c1cccc(NS(=O)(=O)c2ccccc2)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 2/20 0.36
HPGD P15428 2/20 0.34
NR1I2 O75469 2/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
F2 P00734 2/20 0.33
FABP4 P15090 1/20 0.32
ALDH1A1 P00352 3/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
KEAP1 Q14145 1/20 0.31
NFE2L2 Q16236 1/20 0.31
HTR6 P50406 1/20 0.31
PTGES O14684 1/20 0.31
IDH1 O75874 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
PKM P14618 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4828479 0.93 ADRB3 (0.35) ADRB3HPGDNR1I2OPRM1OPRD1
SCHEMBL4891889 0.91 ADRB3 (0.36) ADRB3HPGDNR1I2OPRM1OPRD1
SCHEMBL4778948 0.89 ADRB3 (0.37) ADRB3HPGDNR1I2OPRM1OPRD1
SCHEMBL4837965 0.89 ADRB3 (0.41) ADRB3HPGDNR1I2
SCHEMBL4777051 0.88 ADRB3 (0.37) ADRB3HPGDNR1I2OPRM1OPRD1
SCHEMBL4840597 0.88 ADRB3 (0.37) ADRB3HPGDNR1I2OPRM1OPRD1
SCHEMBL4639769 0.88 ADRB3 (0.36) ADRB3HPGDNR1I2OPRM1OPRD1
SCHEMBL4892190 0.88 NPSR1 (0.38) ADRB3HPGDOPRM1OPRD1ALDH1A1
SCHEMBL4639786 0.87 ADRB3 (0.42) ADRB3HPGDNR1I2OPRM1OPRD1
SCHEMBL4645777 0.86 ADRB3 (0.40) ADRB3HPGDNR1I2OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945304-A2 IMIDAZO-PYRIDINE CONTAINING BETA AGONISTS, METHOD FOR PRODUCING THEM AND THEIR USE AS DRUGS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-07-23 EP disclosed
WO-2007048843-A2 IMIDAZO-PYRIDINE CONTAINING BETA AGONISTS, METHOD FOR PRODUCING THEM AND THEIR USE AS DRUGS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-03 WO disclosed