SCHEMBL4639769

SCHEMBL4639769

CC(C)(CCn1cnc2c(OC(=O)O)cccc21)NCC(OC(=O)C(F)(F)F)c1cccc(NS(=O)(=O)c2ccccc2)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 3/20 0.36
F2 P00734 4/20 0.35
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
HPGD P15428 2/20 0.33
FABP4 P15090 1/20 0.33
NR1I2 O75469 1/20 0.33
ADRB2 P07550 1/20 0.32
ADRB1 P08588 1/20 0.32
ALDH1A1 P00352 2/20 0.32
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
PKM P14618 1/20 0.32
TSHR P16473 1/20 0.32
KEAP1 Q14145 1/20 0.32
NFE2L2 Q16236 1/20 0.32
NPSR1 Q6W5P4 1/20 0.31
KIT P10721 1/20 0.31
EGFR P00533 1/20 0.31
FGFR1 P11362 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4918863 0.91 KEAP1 (0.38) ADRB3F2OPRM1OPRD1HPGD
SCHEMBL4830639 0.88 ADRB3 (0.36) ADRB3F2OPRM1OPRD1HPGD
SCHEMBL4645777 0.87 ADRB3 (0.40) ADRB3F2OPRM1OPRD1HPGD
SCHEMBL4639786 0.87 ADRB3 (0.42) ADRB3F2OPRM1OPRD1HPGD
SCHEMBL4777051 0.86 ADRB3 (0.37) ADRB3F2OPRM1OPRD1HPGD
SCHEMBL4840597 0.86 ADRB3 (0.37) ADRB3F2OPRM1OPRD1HPGD
SCHEMBL4605628 0.85 ADRB3 (0.42) ADRB3F2OPRM1OPRD1HPGD
SCHEMBL4778948 0.85 ADRB3 (0.37) ADRB3F2OPRM1OPRD1HPGD
SCHEMBL4605863 0.85 NR1I2 (0.40) ADRB3OPRM1OPRD1HPGDNR1I2
SCHEMBL4918960 0.84 ADRB3 (0.38) ADRB3F2OPRM1OPRD1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1943229-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-07-16 EP disclosed
WO-2007048842-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-03 WO disclosed