SCHEMBL4833320

SCHEMBL4833320

COC(=O)[C@H](Cc1ccc(-c2ccccc2Oc2ccccc2)cc1)NC(=O)c1cc(Br)ccc1O

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 1/20 0.47
HDAC1 Q13547 5/20 0.45
HDAC6 Q9UBN7 5/20 0.45
TSHR P16473 1/20 0.45
KDR P35968 1/20 0.44
TACR3 P29371 1/20 0.44
ITGA4 P13612 4/20 0.44
ITGB7 P26010 3/20 0.44
ITGB1 P05556 2/20 0.44
CDK2 P24941 2/20 0.43
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
PKM P14618 1/20 0.42
ELANE P08246 2/20 0.42
FFAR4 Q5NUL3 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3996954 0.90 ABCG2 (0.48) ABCG2HDAC1HDAC6TSHRKDR
SCHEMBL3998558 0.90 ABCG2 (0.48) ABCG2HDAC1HDAC6TSHRKDR
SCHEMBL4824030 0.90 PYGL (0.48) HDAC1HDAC6TSHRKDRTACR3
SCHEMBL4824034 0.90 PYGL (0.48) HDAC1HDAC6TSHRKDRTACR3
SCHEMBL4832041 0.90 HDAC1 (0.51) ABCG2HDAC1HDAC6TSHRKDR
SCHEMBL4824867 0.90 HDAC1 (0.51) ABCG2HDAC1HDAC6TSHRKDR
SCHEMBL5927081 0.88 ABCG2 (0.54) ABCG2HDAC1HDAC6TSHRKDR
SCHEMBL5926387 0.88 ABCG2 (0.56) ABCG2TACR3
SCHEMBL5927156 0.88 ABCG2 (0.44) ABCG2HDAC1HDAC6TSHRKDR
SCHEMBL4823477 0.88 HDAC1 (0.56) ABCG2HDAC1HDAC6TSHRKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7459472-B2 Aryl and heteroaryl compounds, compositions, and methods of use TRANSTECH PHARMA, INC. (US) 2008-12-02 US disclosed
US-20050059713-A1 Aryl and heteroaryl compounds, compositions, and methods of use VTVX HOLDINGS I LLC 2005-03-17 US disclosed
WO-2005014534-A1 ARYL AND HETEROARYL COMPOUNDS, COMPOSITIONS, AND METHODS OF USE TRANSTECH PHARMA, INC. (US) 2005-02-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050059713-A1 Aryl and heteroaryl compounds, compositions, and methods of use CYP2F1, CYP3A43, PNPO ABCG2 113/4885HDAC1 1171/4885HDAC6 1063/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.