SCHEMBL483538

SCHEMBL483538

CC(C)(C)OC(=O)N1[C@H](c2cccc(OCc3ccccc3F)c2)CC[C@]12CCCNC2=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN3A Q9NY46 9/20 0.39
F2 P00734 1/20 0.38
F10 P00742 1/20 0.38
BTK Q06187 1/20 0.38
KCNH2 Q12809 7/20 0.38
HPD P32754 1/20 0.37
SPHK2 Q9NRA0 1/20 0.36
SPHK1 Q9NYA1 1/20 0.36
PTPN1 P18031 1/20 0.36
SCN1A P35498 1/20 0.35
SCN4A P35499 1/20 0.35
SCN7A Q01118 1/20 0.35
SCN5A Q14524 1/20 0.35
SCN9A Q15858 1/20 0.35
SCN2A Q99250 1/20 0.35
SCN8A Q9UQD0 1/20 0.35
SCN10A Q9Y5Y9 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2B6 P20813 1/20 0.35
MAOB P27338 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL483225 1.00 SCN3A (0.39) SCN3AF2F10BTKKCNH2
SCHEMBL483533 0.95 F2 (0.39) SCN3AF2F10BTKKCNH2
SCHEMBL484165 0.91 SCN3A (0.48) SCN3ABTKKCNH2SCN1ASCN4A
SCHEMBL483702 0.91 SCN3A (0.48) SCN3ABTKKCNH2SCN1ASCN4A
SCHEMBL2834518 0.89 HPD (0.42) SCN3AF2F10KCNH2HPD
SCHEMBL2835406 0.89 HPD (0.42) SCN3AF2F10KCNH2HPD
SCHEMBL483562 0.86 KCNH2 (0.48) SCN3ABTKKCNH2SCN1ASCN4A
SCHEMBL310836 0.86 KCNH2 (0.48) SCN3ABTKKCNH2SCN1ASCN4A
SCHEMBL483745 0.85 BTK (0.40) SCN3AF2F10BTKKCNH2
SCHEMBL2832474 0.83 KCNH2 (0.42) SCN3AF2F10KCNH2HPD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8153623-B2 Compounds Convergence Pharmaceuticals Limited (GB) 2012-04-10 US disclosed
EP-1934176-B1 QUATERNARY ALPHA-AMINOCARBOXAMIDE DERIVATIVES AS MODULATORS OF VOLTAGE-GATED SODIUM CHANNELS GLAXO GROUP LTD (GB) 2012-02-01 EP disclosed