SCHEMBL4836388

SCHEMBL4836388

COc1ccc(-c2[nH]nnc2-c2ccc(OC)c(OC)c2OC)cc1NC(=O)CCC(=O)O

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.42
LTB4R Q15722 2/20 0.39
HPGD P15428 2/20 0.38
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
CYP1A2 P05177 1/20 0.38
HSD17B10 Q99714 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
MAPT P10636 3/20 0.38
KMT2A Q03164 1/20 0.38
CYP2C9 P11712 1/20 0.37
TSHR P16473 2/20 0.37
POLB P06746 1/20 0.37
LMNA P02545 1/20 0.36
PKM P14618 1/20 0.36
GAA P10253 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL412790 0.89 NPSR1 (0.41) NPSR1LTB4RHPGDALDH1A1SMN1; SMN2
SCHEMBL413515 0.83 EGFR (0.43) NPSR1LTB4RKMT2APOLBGAA
SCHEMBL410256 0.83 NPC1 (0.40) NPSR1LTB4RALDH1A1SMN1; SMN2MAPT
SCHEMBL13041260 0.82 NPSR1 (0.50) NPSR1LTB4RHPGDALDH1A1KDM4E
SCHEMBL3300296 0.79 NPSR1 (0.43) NPSR1LTB4RHPGDALDH1A1KDM4E
Hydrochloric Acid SCHEMBL4629522 0.79 NPSR1 (0.41) NPSR1LTB4RHPGDALDH1A1KDM4E
Hydrochloric Acid SCHEMBL411516 0.78 NPSR1 (0.42) NPSR1LTB4RHPGDALDH1A1KDM4E
SCHEMBL14401731 0.77 NPSR1 (0.39) NPSR1LTB4RHPGDALDH1A1KDM4E
SCHEMBL3303665 0.77 NPC1 (0.39) NPSR1HPGDALDH1A1KDM4ECYP1A2
SCHEMBL411454 0.76 POLB (0.43) NPSR1LTB4RHPGDALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919881-A1 1, 2, 3 -TRIAZOLES INHIBITORS OF TUBULIN POLYMERIZATION FOR THE TREATMENT OF POLIFERATIVE DISORDERS Synta Pharmaceuticals Corporation (US) 2008-05-14 EP disclosed
WO-2007014198-A1 1, 2, 3 -TRIAZOLES INHIBITORS OF TUBULIN POLYMERIZATION FOR THE TREATMENT OF POLIFERATIVE DISORDERS SYNTA PHARMACEUTICALS CORP. (US) 2007-02-01 WO disclosed