SCHEMBL483699

SCHEMBL483699

CN1[C@@H](c2ccc(OCc3ccccc3F)cc2)CCC[C@H]1C(=O)O

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.72
SCN3A Q9NY46 7/20 0.62
FFAR2 O15552 1/20 0.52
SCN9A Q15858 2/20 0.50
SCN1A P35498 1/20 0.50
SCN4A P35499 1/20 0.50
SCN7A Q01118 1/20 0.50
SCN5A Q14524 1/20 0.50
SCN2A Q99250 1/20 0.50
SCN8A Q9UQD0 1/20 0.50
SCN10A Q9Y5Y9 1/20 0.50
MAOB P27338 3/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2B6 P20813 1/20 0.49
CYP2C19 P33261 1/20 0.49
LPAR1 Q92633 2/20 0.46
LPAR5 Q9H1C0 2/20 0.46
PARP15 Q460N3 1/20 0.46
PARP14 Q460N5 1/20 0.46
PARP10 Q53GL7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1093299 1.00 KCNH2 (0.72) KCNH2SCN3AFFAR2SCN9ASCN1A
SCHEMBL310295 0.94 KCNH2 (0.82) KCNH2SCN3AFFAR2SCN9ASCN1A
SCHEMBL310303 0.94 KCNH2 (0.82) KCNH2SCN3AFFAR2SCN9ASCN1A
SCHEMBL2836386 0.87 KCNH2 (0.58) KCNH2SCN3AFFAR2SCN9ASCN1A
SCHEMBL2839975 0.84 KCNH2 (1.00) KCNH2SCN3AFFAR2SCN9ASCN1A
SCHEMBL17873393 0.83 KCNH2 (0.66) KCNH2SCN3AFFAR2SCN9ASCN1A
SCHEMBL24279500 0.83 KCNH2 (0.79) KCNH2SCN3AFFAR2SCN9ASCN1A
Hydrochloric Acid SCHEMBL2836853 0.83 KCNH2 (0.98) KCNH2SCN3AFFAR2SCN9ASCN1A
SCHEMBL2835344 0.82 KCNH2 (0.77) KCNH2SCN3AFFAR2SCN9ASCN1A
Hydrochloric Acid SCHEMBL2837163 0.81 KCNH2 (0.76) KCNH2SCN3AFFAR2SCN9ASCN1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8153623-B2 Compounds Convergence Pharmaceuticals Limited (GB) 2012-04-10 US disclosed
EP-1934176-B1 QUATERNARY ALPHA-AMINOCARBOXAMIDE DERIVATIVES AS MODULATORS OF VOLTAGE-GATED SODIUM CHANNELS GLAXO GROUP LTD (GB) 2012-02-01 EP disclosed