SCHEMBL483726

SCHEMBL483726

O=CCc1ccc(-c2ccc(F)nc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.44
CYP2B6 P20813 3/20 0.44
CYP2E1 P05181 1/20 0.44
CNR1 P21554 2/20 0.38
CHRM5 P08912 1/20 0.38
CYP11B2 P19099 2/20 0.38
CYP3A4 P08684 3/20 0.38
CYP2C19 P33261 2/20 0.38
DHODH Q02127 1/20 0.38
JAK2 O60674 1/20 0.37
RET P07949 1/20 0.37
KDR P35968 1/20 0.37
GSK3A P49840 1/20 0.37
RPS6KA3 P51812 1/20 0.37
LIMK1 P53667 1/20 0.37
MAP2K1 Q02750 1/20 0.37
DYRK1A Q13627 1/20 0.37
MAPK14 Q16539 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
ALK Q9UM73 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL114699 0.84 CYP11B1 (0.43) CYP2A6CYP2B6CYP2E1CYP11B2CYP11B1
SCHEMBL12917647 0.78 MKNK1 (0.51) CNR1DYRK1ADYRK1BCYP1A2
SCHEMBL12496644 0.77 HRH3 (0.56) CYP2A6CYP2B6CYP2E1CYP11B2CYP3A4
SCHEMBL9158239 0.77 CYP2A6 (0.47) CYP2A6CYP2B6CYP2E1CNR1CHRM5
SCHEMBL9156751 0.77 CYP2A6 (0.47) CYP2A6CYP2B6CYP2E1CNR1CHRM5
SCHEMBL3392101 0.77 HRH3 (0.43)
SCHEMBL26104326 0.77 CYP2A6 (0.64) CYP2A6CYP2B6CYP2E1CYP11B2CYP3A4
SCHEMBL17423600 0.76 MAOB (0.48)
Hydrochloric Acid SCHEMBL21352581 0.75 HRH3 (0.41) CYP1A2
SCHEMBL6851863 0.74 HDAC4 (0.40) CYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411057-A2 IMAGING AGENTS FOR DETECTING NEUROLOGICAL DISORDERS Siemens Medical Solutions USA, Inc. (US) 2012-02-01 EP disclosed
WO-2010111303-A2 IMAGING AGENTS FOR DETECTING NEUROLOGICAL DISORDERS SIEMENS MEDICAL SOLUTIONS USA, INC. (US) 2010-09-30 WO disclosed