SCHEMBL9156751

SCHEMBL9156751

CCc1ccc(-c2ccc(-c3ccc(F)nc3)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.47
CYP2B6 P20813 3/20 0.47
CYP2E1 P05181 1/20 0.47
CYP3A4 P08684 3/20 0.43
CYP2C19 P33261 2/20 0.43
METAP2 P50579 1/20 0.42
CYP11B2 P19099 2/20 0.40
CHRM5 P08912 1/20 0.40
USP1 O94782 1/20 0.39
WDR48 Q8TAF3 1/20 0.39
EGLN1 Q9GZT9 1/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
CNR1 P21554 2/20 0.38
CYP11B1 P15538 1/20 0.38
MMP2 P08253 1/20 0.38
MMP9 P14780 1/20 0.38
MMP13 P45452 1/20 0.38
GRIN1 Q05586 2/20 0.37
GRIN2B Q13224 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9158239 1.00 CYP2A6 (0.47) CYP2A6CYP2B6CYP2E1CYP3A4CYP2C19
SCHEMBL9154340 0.87 NPC1 (0.40) CYP2A6CYP2B6CYP2E1CYP3A4CYP2C19
SCHEMBL9156341 0.85 CYP2A6 (0.44) CYP2A6CYP2B6CYP2E1CYP3A4CYP2C19
SCHEMBL9158742 0.85 CYP2A6 (0.44) CYP2A6CYP2B6CYP2E1CYP3A4CYP2C19
SCHEMBL9156736 0.84 PDE3B (0.42) CYP2A6CYP2B6CYP2E1CYP3A4CYP2C19
SCHEMBL357013 0.83
SCHEMBL9154247 0.83 GRM5 (0.47) CYP2A6METAP2EGLN1
SCHEMBL9766634 0.82 MAPT (0.48) CYP3A4CHRM5LMNATP53
SCHEMBL15304176 0.82 RAB9A (0.58) CYP2A6CYP2B6CYP2E1CYP3A4CYP2C19
SCHEMBL9161126 0.82 RARB (0.47) CYP2A6CYP2B6CYP2E1CYP3A4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445248-B1 PYRIDINE DERIVATIVES MERCK PATENT GMBH (DE) 1995-03-08 EP disclosed
US-5205962-A Stable liquid crystals MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1993-04-27 US disclosed