SCHEMBL4839137

SCHEMBL4839137

CC(=O)N1CCN(C(=O)c2cc3ncnc(NCCc4nc5cc(Cl)ccc5[nH]4)c3cc2Cl)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.42
CDK1 P06493 6/20 0.40
HTT P42858 3/20 0.38
CLK1 P49759 1/20 0.38
NR2F2 P24468 1/20 0.38
CCNC P24863 1/20 0.38
CDK8 P49336 1/20 0.38
MAP4K2 Q12851 1/20 0.38
HASPIN Q8TF76 1/20 0.38
CDK19 Q9BWU1 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
MAPK8 P45983 3/20 0.37
MAPK10 P53779 3/20 0.37
HRH4 Q9H3N8 1/20 0.37
F9 P00740 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
RHEB Q15382 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4844553 0.88 GAA (0.42) CDK1HTTNR2F2HDAC1HDAC8
SCHEMBL4148481 0.84 CDK1 (0.43) CDK1MAPK8MAPK10HRH4
SCHEMBL4150594 0.82 CLK1 (0.38) LMNACDK1CLK1HRH4CNR1
SCHEMBL4839125 0.77 LMNA (0.40) LMNACLK1HRH4
SCHEMBL4841553 0.76 CNR1 (0.36) CDK1HDAC1HDAC8HDAC6MAPK8
SCHEMBL4150728 0.76 KDM4E (0.40) LMNAHTTHDAC1HDAC8HDAC6
SCHEMBL4156270 0.75 HRH4 (0.36) LMNACDK1MAPK8MAPK10HRH4
SCHEMBL2995838 0.75 HRH4 (0.40) CDK1HRH4CNR1CNR2
SCHEMBL2995841 0.75 HRH4 (0.40) CDK1HRH4CNR1CNR2
SCHEMBL4841881 0.75 HRH4 (0.35) CDK1HDAC1HDAC8HDAC6HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7429597-B2 Substituted nitrogen-containing heterobicycles, the preparation thereof and their use as pharmaceutical compositions BOEHRINGER INGELHEIM PHARMA GMBH & CO., KG (DE) 2008-09-30 US claimed