SCHEMBL48395

SCHEMBL48395

Nc1ccn(O)c(=O)n1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11894064 0.74
SCHEMBL25378286 0.74
SCHEMBL22016090 0.74
SCHEMBL12096477 0.74 FGFR1 (0.39)
SCHEMBL1179743 0.74 PDE3A (0.36)
SCHEMBL5985575 0.73
SCHEMBL4492972 0.73
SCHEMBL8944773 0.73
SCHEMBL7876669 0.73
SCHEMBL19692381 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 173 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025038971-A1 OLIGONUCLEOTIDES CONTAINING A LIGAND AT A NUCLEOBASE, 2' POSITION, OR 3' POSITION ADARX PHARMACEUTICALS, INC. (US) 2025-02-20 WO claimed
CN-118086264-A Cytidine deaminase immobilization based on T4 phage-bound magnetic bead composite material 江苏海洋大学 2024-05-28 CN claimed
CN-117881403-A Thionucleosides as antiviral agents 爱莫里大学 2024-04-12 CN claimed
CN-117858711-A Nucleoside and nucleotide analogs as antiviral agents 爱莫里大学 2024-04-09 CN claimed
CN-117512078-A Single primer to double primer amplicon conversion 西格马-奥尔德里奇有限责任公司 2024-02-06 CN claimed
US-20230357168-A1 CARBOBICYCLIC NUCLEOSIDES FOR TREATMENT OF VIRAL INFECTION UNIV HONG KONG CHINESE (CN) 2023-11-09 US claimed
CN-109804083-B Single primer to double primer amplicon conversion 西格马-奥尔德里奇有限责任公司 2023-11-03 CN claimed
WO-2023198181-A1 CARBOBICYCLIC NUCLEOSIDES FOR TREATMENT OF VIRAL INFECTION THE CHINESE UNIVERSITY OF HONG KONG (CN) 2023-10-19 WO claimed
US-20220315972-A1 SINGLE PRIMER TO DUAL PRIMER AMPLICON SWITCHING SIGMA ALDRICH CO LLC (US) 2022-10-06 US claimed
US-11390913-B2 Single primer to dual primer amplicon switching SIGMA-ALDRICH CO. LLC (US) 2022-07-19 US claimed
US-20210332078-A1 COMPOSITIONS AND METHODS FOR NUCLEIC ACID AMPLIFICATION Twist Bioscience Corporation 2021-10-28 US claimed
EP-3516075-A1 SINGLE PRIMER TO DUAL PRIMER AMPLICON SWITCHING Sigma-Aldrich Co., LLC (US) 2019-07-31 EP claimed
US-20190211386-A1 SINGLE PRIMER TO DUAL PRIMER AMPLICON SWITCHING SIGMA-ALDRICH CO. LLC 2019-07-11 US claimed
CN-109804083-A Single primer to double primer amplicon conversion 西格马-奥尔德里奇有限责任公司 2019-05-24 CN claimed
WO-2018057846-A1 SINGLE PRIMER TO DUAL PRIMER AMPLICON SWITCHING SIGMA-ALDRICH CO, LLC (US) 2018-03-29 WO claimed
US-20160333340-A1 COMPOSITIONS AND METHODS FOR NUCLEIC ACID AMPLIFICATION Twist Bioscience Corporation 2016-11-17 US claimed
WO-2016183100-A1 COMPOSITIONS AND METHODS FOR NUCLEIC ACID AMPLIFICATION Twist Bioscience Corporation (US) 2016-11-17 WO claimed
EP-2271653-A2 NOVEL METHOD FOR PREPARING OLIGONUCLEOTIDES COMPRISING A 5' -PHOSPHATE MONOESTER OR 5' -THIOPHOSPHATE MONOESTER END Université Joseph Fourier (FR) 2011-01-12 EP claimed
WO-2009138614-A2 NOVEL METHOD FOR PREPARING OLIGONUCLEOTIDES COMPRISING A 5’-PHOSPHATE MONOESTER OR 5’-THIOPHOSPHATE MONOESTER END UNIVERSITE JOSEPH FOURIER (FR) 2009-11-19 WO claimed
WO-2008033432-A2 IMMUNE MODULATION BY CHEMICALLY MODIFIED RIBONUCLEOSIDES AND OLIGORIBONUCLEOTIDES COLEY PHARMACEUTICAL GROUP, INC. (US) 2008-03-20 WO claimed