SCHEMBL4840144

SCHEMBL4840144

CCCc1nc(N)nc2ccc(-c3cccc(OCC#N)c3)nc12.CCCc1nc(N)nc2ccc(-c3ccccc3OCC#N)nc12

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAOB P27338 8/20 0.40
MAOA P21397 4/20 0.40
MAP4K4 O95819 6/20 0.39
ALOX5AP P20292 2/20 0.38
FEN1 P39748 2/20 0.38
DHFR P00374 3/20 0.35
PFKFB3 Q16875 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4114833 0.92 MAOB (0.46) MAOBMAOAMAP4K4DHFRPFKFB3
SCHEMBL4102014 0.90 MAOB (0.44) MAOBMAOAALOX5APFEN1DHFR
SCHEMBL4104502 0.80 MAOB (0.41) MAOBMAOADHFR
SCHEMBL4097650 0.80 MAOB (0.46) MAOBMAOAMAP4K4DHFRPFKFB3
SCHEMBL4113326 0.78 MAP4K4 (0.56) MAP4K4DHFR
SCHEMBL4096455 0.77 MAOB (0.49) MAOBMAOAMAP4K4PFKFB3
SCHEMBL4108022 0.77 MAOB (0.44) MAOBMAOAALOX5APFEN1DHFR
SCHEMBL4113347 0.76 MAOB (0.45) MAOBMAOAALOX5APFEN1
SCHEMBL4107331 0.76 TLR4 (0.47) DHFR
SCHEMBL4097587 0.75 CTSS (0.51) MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009076-A2 SUBSTITUTED PYRIDO(3,2-D)PYRIMIDINES AND PHARMACEUTICAL COMPOSITIONS FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO claimed