SCHEMBL4840985

SCHEMBL4840985

C=CCn1cc(Br)nc1CBr

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CSNK2A2 P19784 1/20 0.35
CSNK2B P67870 1/20 0.35
CSNK2A1 P68400 1/20 0.35
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33
ADORA1 P30542 1/20 0.33
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
PDE4B Q07343 1/20 0.30
PDE4D Q08499 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23214483 0.73 CYP3A4 (0.40) CSNK2A2CSNK2BCSNK2A1ADORA2AADORA2B
SCHEMBL23214023 0.67 CYP1A2 (0.36) ADORA2AADORA2BCYP1A2CYP3A4CYP2D6
SCHEMBL374956 0.64 CYP1A2 (0.32) CYP1A2CYP3A4CYP2D6PDE4BPDE4D
SCHEMBL4851130 0.63 ADORA2B (0.36) CSNK2A2CSNK2BCSNK2A1ADORA3ADORA2A
SCHEMBL6001890 0.63 CYP19A1 (0.42) ADORA2BCYP1A2CYP3A4CYP2D6
SCHEMBL14938360 0.63 MEN1 (0.31) CYP1A2CYP3A4CYP2D6PDE4BPDE4D
Iodide SCHEMBL3468594 0.63 CYP1A2 (0.31) CYP1A2CYP3A4CYP2D6PDE4BPDE4D
SCHEMBL9038600 0.63 CYP1A2 (0.31) CYP1A2CYP3A4CYP2D6PDE4BPDE4D
Hydrochloric Acid SCHEMBL3260796 0.63 CYP1A2 (0.31) CYP1A2CYP3A4CYP2D6PDE4BPDE4D
SCHEMBL11167293 0.59 CYP3A4 (0.38) ADORA2AADORA2BCYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008033455-A2 BIPHENYL AND HETEROARYL PHENYL DERIVATIVES AS PROTEIN TYROSINE PHOSPHATASES INHIBITORS THE INSTITUTES FOR PHARMACEUTICAL DISCOVERY, LLC (US) 2008-03-20 WO disclosed