SCHEMBL4846612

SCHEMBL4846612

CC(=O)c1cccc(OCCN(C)C)c1

nearest known ligand 0.63

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.63
CHRNB2 P17787 2/20 0.62
CHRNA4 P43681 2/20 0.62
KDM4E B2RXH2 5/20 0.61
ALDH1A1 P00352 3/20 0.61
LMNA P02545 1/20 0.61
THRA P10827 1/20 0.58
THRB P10828 1/20 0.58
MAOB P27338 7/20 0.57
MAOA P21397 2/20 0.54
KMT2A Q03164 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6623073 0.88 KMT2A (0.69) ESR1CHRNB2CHRNA4KDM4EALDH1A1
SCHEMBL5974513 0.87 MAOB (0.68) ALDH1A1MAOBMAOAKMT2ASMN1; SMN2
Hydrochloric Acid SCHEMBL8702528 0.86 KMT2A (0.68) ESR1CHRNB2CHRNA4KDM4EALDH1A1
SCHEMBL3652803 0.86 ESR1 (0.61) ESR1CHRNB2CHRNA4KDM4EALDH1A1
SCHEMBL4638666 0.85 ESR1 (0.67) ESR1CHRNB2CHRNA4KDM4EALDH1A1
SCHEMBL8126769 0.85 ESR1 (0.60) ESR1CHRNB2CHRNA4KDM4EALDH1A1
SCHEMBL14511273 0.83 MAPT (0.53) ESR1CHRNB2CHRNA4KDM4EALDH1A1
SCHEMBL7632070 0.82 ESR1 (0.57) ESR1CHRNB2CHRNA4KDM4EALDH1A1
SCHEMBL4315663 0.82 MAOB (0.62) ALDH1A1MAOBMAOAKMT2ASMN1; SMN2
SCHEMBL1436064 0.82 KMT2A (0.76) MAOBMAOAKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed
EP-1515940-A2 AMINOALKOXY-FUNCTIONAL CHALCONES Lica Pharmaceuticals A/S (DK) 2005-03-23 EP disclosed
WO-2003097574-A2 AMINOALKOXY-FUNCTIONAL CHALCONES LICA PHARMACEUTICALS A/S (DK) 2003-11-27 WO disclosed