SCHEMBL4846787

SCHEMBL4846787

CN(C)CCOc1ccc(C(=O)C=Cc2ccc(Cl)cc2Cl)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 6/20 0.61
ACHE P22303 6/20 0.61
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C19 P33261 1/20 0.51
MAPT P10636 3/20 0.50
LMNA P02545 3/20 0.50
DPP4 P27487 2/20 0.50
BLM P54132 1/20 0.50
PMP22 Q01453 1/20 0.50
HPGD P15428 1/20 0.50
MAOB P27338 2/20 0.49
HRH3 Q9Y5N1 1/20 0.49
ALDH1A1 P00352 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
NPC1 O15118 1/20 0.48
POLB P06746 1/20 0.48
RAB9A P51151 1/20 0.48
KDM4E B2RXH2 2/20 0.47
PKM P14618 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4849641 0.88 KDM4E (0.56) BCHEACHEMAPTLMNAMAOB
SCHEMBL4846156 0.84 KDM4E (0.46) BCHEACHECYP1A2CYP3A4CYP2C19
SCHEMBL29181781 0.84 DPP4 (0.52) MAPTLMNADPP4HPGDMAOB
SCHEMBL3687525 0.81 MAPT (0.50) CYP1A2CYP2C19MAPTLMNAHPGD
SCHEMBL1225611 0.80 MAOB (0.71) CYP1A2CYP3A4CYP2C19MAPTLMNA
SCHEMBL1225612 0.80 MAOB (0.71) CYP1A2CYP3A4CYP2C19MAPTLMNA
SCHEMBL4846128 0.80 PTPN5 (0.54) BCHEACHEMAPTLMNAHPGD
SCHEMBL4852869 0.80 KDM4E (0.46) BCHEACHECYP1A2CYP3A4CYP2C19
SCHEMBL4846138 0.80 KDM4E (0.46) BCHEACHECYP1A2CYP3A4CYP2C19
SCHEMBL5915668 0.80 MAPT (0.53) CYP1A2CYP2C19MAPTLMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US claimed
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed