SCHEMBL4849684

SCHEMBL4849684

CCN(CC)CCOc1ccc(-c2ccccc2C)cc1C(=O)/C=C/c1ccccc1CN(C)C

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 2/20 0.44
MCHR1 Q99705 4/20 0.40
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.39
MAOB P27338 7/20 0.38
BCHE P06276 2/20 0.38
ACHE P22303 2/20 0.38
HPGD P15428 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MAOA P21397 6/20 0.37
APP P05067 4/20 0.37
PTPN11 Q06124 1/20 0.37
AR P10275 1/20 0.36
DRD2 P14416 1/20 0.36
DRD1 P21728 1/20 0.36
DRD3 P35462 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4850218 1.00 SLC6A9 (0.44) SLC6A9MCHR1KDM4EALDH1A1LMNA
SCHEMBL4845305 0.95 MAOB (0.42) SLC6A9MAOBBCHEACHEMAOA
SCHEMBL4852558 0.95 MAOB (0.42) SLC6A9MAOBBCHEACHEMAOA
SCHEMBL4847435 0.93 SLC6A9 (0.46) SLC6A9MCHR1KDM4EALDH1A1BCHE
SCHEMBL4853568 0.93 SLC6A9 (0.46) SLC6A9MCHR1KDM4EALDH1A1BCHE
SCHEMBL4849688 0.90 SLC6A9 (0.41) SLC6A9MCHR1KDM4EALDH1A1LMNA
SCHEMBL4854469 0.90 SLC6A9 (0.43) SLC6A9KDM4EALDH1A1BCHEACHE
SCHEMBL4856457 0.90 SLC6A9 (0.43) SLC6A9KDM4EALDH1A1BCHEACHE
SCHEMBL4847208 0.89 SLC6A9 (0.43) SLC6A9MCHR1KDM4EALDH1A1LMNA
SCHEMBL4852352 0.89 SLC6A9 (0.43) SLC6A9MCHR1KDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed