SCHEMBL4852282

SCHEMBL4852282

COc1ccc(C(=O)C=Cc2ccc(OCCN(C)C)cc2)c(OC)c1OC

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TUBB1 Q9H4B7 3/20 0.58
BCHE P06276 3/20 0.57
ACHE P22303 3/20 0.57
MCL1 Q07820 3/20 0.54
CYP3A4 P08684 1/20 0.53
CYP1A1 P04798 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP1B1 Q16678 1/20 0.52
MAOB P27338 1/20 0.52
ABCG2 Q9UNQ0 3/20 0.51
MAPT P10636 2/20 0.50
MEN1 O00255 1/20 0.50
USP2 O75604 1/20 0.50
MAPK1 P28482 1/20 0.50
KMT2A Q03164 1/20 0.50
TLR9 Q9NR96 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
TNFRSF1A P19438 1/20 0.50
APP P05067 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1425149 0.87 TUBB1 (0.61) TUBB1MCL1CYP3A4CYP1A1CYP1A2
SCHEMBL1425154 0.87 TUBB1 (0.61) TUBB1MCL1CYP3A4CYP1A1CYP1A2
SCHEMBL4846963 0.87 TUBB1 (0.56) TUBB1BCHEACHEMCL1CYP3A4
SCHEMBL4851201 0.85 ABCG2 (0.73) BCHEACHEABCG2MAPTMEN1
SCHEMBL4845554 0.85 ABCG2 (0.73) BCHEACHEABCG2MAPTMEN1
SCHEMBL15756405 0.85 TUBB1 (0.64) TUBB1MCL1CYP3A4CYP1A1CYP1A2
SCHEMBL15756404 0.85 TUBB1 (0.64) TUBB1MCL1CYP3A4CYP1A1CYP1A2
SCHEMBL5915484 0.84 TUBB1 (0.60) TUBB1MCL1CYP3A4CYP1A1CYP1A2
SCHEMBL15304531 0.83 TUBB1 (0.71) TUBB1MCL1CYP3A4CYP1A1CYP1A2
SCHEMBL4849390 0.82 ALDH1A1 (0.52) TUBB1BCHECYP1A1CYP1A2CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US claimed
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed