SCHEMBL4853145

SCHEMBL4853145

[CH2]C1CCN(C(=O)Cc2ccncc2)C(C(N)=O)C1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 10/20 0.40
PARP1 P09874 1/20 0.38
FNTA P49354 2/20 0.38
FNTB P49356 2/20 0.38
SIGMAR1 Q99720 1/20 0.36
OPRK1 P41145 1/20 0.35
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30874862 0.82 CYP19A1 (0.47) CYP19A1SMN1; SMN2
SCHEMBL4701608 0.77 CYP19A1 (0.42) CYP19A1PARP1FNTAFNTBSIGMAR1
SCHEMBL4700677 0.75 SYK (0.39) LMNA
SCHEMBL30874874 0.68 VNN1 (0.44)
SCHEMBL474918 0.68 DPP4 (0.57) ALDH1A1HPGD
SCHEMBL2177077 0.68 DPP4 (0.57) ALDH1A1HPGD
SCHEMBL30874798 0.68 VNN1 (0.62) PARP1FNTAFNTBSIGMAR1ALDH1A1
SCHEMBL4701611 0.67 FNTA (0.53) CYP19A1FNTAFNTBALDH1A1LMNA
SCHEMBL4705648 0.66 FNTA (0.49) FNTAFNTBALDH1A1LMNA
SCHEMBL30874864 0.66 VNN1 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7432379-B2 Substituted pyrazole derivatives and related compounds as bradykinin B1 receptor antagonists ELAN PHARMACEUTICALS, INC. (US) 2008-10-07 US claimed