SCHEMBL4856632

SCHEMBL4856632

Cc1cc(C)cc(-c2ccc(OCCN(C)C)c(C(=O)/C=C/c3cccc(Br)c3)c2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 2/20 0.44
ALDH1A1 P00352 3/20 0.43
LMNA P02545 3/20 0.43
KDM4E B2RXH2 2/20 0.43
BCHE P06276 2/20 0.42
ACHE P22303 2/20 0.42
MAOB P27338 3/20 0.41
MAOA P21397 1/20 0.41
MAPT P10636 2/20 0.41
MEN1 O00255 1/20 0.41
POLB P06746 1/20 0.41
XBP1 P17861 1/20 0.41
ALOX12 P18054 1/20 0.41
RECQL P46063 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CYP2D6 P10635 2/20 0.40
CYP1B1 Q16678 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4857214 1.00 SYK (0.44) SYKALDH1A1LMNAKDM4EBCHE
SCHEMBL4853507 0.90 MAOA (0.44) SYKBCHEACHEMAOBMAOA
SCHEMBL4857314 0.90 MAOA (0.44) SYKBCHEACHEMAOBMAOA
SCHEMBL4857397 0.89 SYK (0.45) SYKALDH1A1LMNAKDM4EBCHE
SCHEMBL4849917 0.89 SYK (0.45) SYKALDH1A1LMNAKDM4EBCHE
SCHEMBL4853732 0.89 BCHE (0.54) SYKBCHEACHESLC6A9
SCHEMBL4854231 0.89 BCHE (0.54) SYKBCHEACHESLC6A9
SCHEMBL4853337 0.89 SYK (0.44) SYKLMNAKDM4EBCHEACHE
SCHEMBL4846158 0.88 BCHE (0.41) SYKBCHEACHEMAOBSLC6A9
SCHEMBL4854696 0.88 BCHE (0.41) SYKBCHEACHEMAOBSLC6A9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed