SCHEMBL4859342

SCHEMBL4859342

COC(=O)c1cnc(N2CCN(C(c3ccccc3C(F)(F)F)C(F)(F)F)CC2)s1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCD O00767 8/20 0.51
HRH3 Q9Y5N1 2/20 0.47
OGA O60502 4/20 0.41
HDAC3 O15379 3/20 0.40
HDAC4 P56524 3/20 0.40
HDAC1 Q13547 3/20 0.40
HDAC7 Q8WUI4 3/20 0.40
HDAC2 Q92769 3/20 0.40
HDAC10 Q969S8 3/20 0.40
HDAC11 Q96DB2 3/20 0.40
HDAC8 Q9BY41 3/20 0.40
HDAC6 Q9UBN7 3/20 0.40
HDAC9 Q9UKV0 3/20 0.40
HDAC5 Q9UQL6 3/20 0.40
CRBN Q96SW2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25348 0.79 SCD (0.80) SCDHDAC3HDAC4HDAC1HDAC7
SCHEMBL4087735 0.79 SCD (0.77) SCD
SCHEMBL4814710 0.76 OGA (0.57) HRH3OGA
SCHEMBL472984 0.75 SCD (0.78) SCDHRH3
SCHEMBL3159765 0.72 HRH3 (0.54) HRH3OGAHDAC3HDAC4HDAC1
SCHEMBL2946807 0.72 SCD (0.79) SCDHRH3
SCHEMBL2945498 0.72 SCD (0.79) SCDHRH3
SCHEMBL4807896 0.71 HDAC3 (0.74) SCDHRH3HDAC3HDAC4HDAC1
SCHEMBL4804346 0.71 ALDH1A1 (0.61) SCDHRH3HDAC3HDAC4HDAC1
SCHEMBL20176409 0.71 HRH3 (0.57) HRH3OGAHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902051-A1 AZACYCLOHEXANE DERIVATIVES AS INHIBITORS OF STEAROYL-COENZYME A DELTA-9 DESATURASE Merck Frosst Canada Ltd. (CA) 2008-03-26 EP disclosed
WO-2006130986-A1 AZACYCLOHEXANE DERIVATIVES AS INHIBITORS OF STEAROYL-COENZYME A DELTA-9 DESATURASE MERCK FROSST CANADA LTD. (CA) 2006-12-14 WO disclosed